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(2S)-2-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}propanamide
methyl 3-[2-(2,3-difluorophenyl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-methyl-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}but-2-en-1-one
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}propane-1,3-diol
(2-ethoxy-5-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}phenyl)methanol
4-(propan-2-yl)-6-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]pyrimidin-2-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-[(4-fluorophenyl)methyl]-4-[3-(methylsulfanyl)propyl]morpholine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-(2-fluorophenyl)-4-(2-methylphenyl)-1,4-diazepane-1-carboxamide
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-3-(1H-pyrazol-1-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
1-(2-{[cyclohexyl(methyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
3-(1-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
{4-[(4-methoxyphenyl)methyl]-1-(quinolin-8-ylmethyl)piperidin-4-yl}methanol
1-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-3-phenylpropan-1-ol
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][2-(4-chlorophenyl)ethyl](pyridin-4-ylmethyl)amine
[(2-{[5-(methanesulfonylmethyl)pyridin-2-yl]oxy}phenyl)methyl]dimethylamine
2-(2-hydroxyethyl)-9-[2-(2-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperazine-1-sulfonamide
(3S,4S)-4-cyclopropyl-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-(2-{[(3-cyano-4-methoxyphenyl)carbamoyl]amino}ethyl)acetamide
2-(5-acetylthiophen-3-yl)-1-[2-(furan-2-yl)azepan-1-yl]ethan-1-one
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-cyclohexyl-1H-pyrazol-5-yl)acetamide
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)methanesulfonamide
(1S,3R)-3-amino-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}cyclopentane-1-carboxamide
4-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-2-one
3-ethyl-1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
(3S)-4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,3-dimethylpiperazin-2-one
4-[4-(3-methoxypiperidin-1-yl)pyridine-2-carbonyl]morpholine
5-(methoxymethyl)-N-{4-[5-methyl-4-({spiro[2.4]heptan-1-ylformamido}methyl)-1,3-oxazol-2-yl]phenyl}thiophene-2-carboxamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-[2-(furan-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-1-methyl-1H-1,3-benzodiazole
methyl (2S)-2-({1-[4-(cyclopentylcarbamoyl)phenyl]piperidin-4-yl}amino)-2-phenylacetate
4-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
5-(2-chlorophenyl)-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]furan-2-carboxamide
N-cyclopropyl-1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3-(2-methylpropyl)-1,2-oxazole
3-ethyl-8-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({3-methyl-7-[4-(pyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
[1-(4-amino-6,7-dimethoxyquinazolin-2-yl)-3-propylpiperidin-3-yl]methanol
5-[4-(benzenesulfonyl)piperazine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-decahydroisoquinoline
1-{2-[3-(3-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}azepan-2-one
2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]ethan-1-amine
1-methyl-3-(2-phenylethyl)-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione