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1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-methoxybenzoyl)piperazine
ethyl 1-(2-fluorobenzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
(3aS,6aR)-5-[(2-fluorophenyl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-{3-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-[(3-methoxyphenyl)methyl]-3-[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]propanamide
3-{1-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
3-methoxy-N,4-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
3-({7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)benzonitrile
N-[(3R,4R)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
2-cyclopropyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
2,6,8-trimethyl-4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
1-(1-{4-[1-(cyclopropylmethyl)-1H-pyrazol-4-yl]phenyl}ethyl)piperidine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-(thiophen-3-ylmethyl)benzamide
1-{1-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperidin-4-yl}-1,4-diazepan-5-one
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(4-fluoro-2-methoxyphenyl)methyl](2-methoxyethyl)amine
1-benzyl-N-(3-ethoxypropyl)-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-[3-(prop-2-en-1-yloxy)benzoyl]-1,4-diazepan-6-yl}oxy)acetamide
3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-methyl-1-[(2-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
5-(4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-cyclopentanecarbonyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylpiperidine-4-carboxamide
3-{5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2,5,6-trimethylpyrimidin-4-amine
N-methyl-N-[2-(2-methylphenyl)-1-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]ethyl]-2-(1H-pyrazol-1-yl)acetamide
1-(1-benzofuran-3-carbonyl)-4,4-difluoropiperidine
6-methyl-2-(morpholin-4-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
6-tert-butyl-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-oxo-2,3-dihydropyrimidine-4-carboxamide
4-[(4-methylphenyl)sulfanyl]-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
N-[(3,4-dimethoxyphenyl)methyl]-2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}acetamide
methyl 3-(5-methoxy-5-oxopentanoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 4-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(2S,4S)-1-benzyl-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
3-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4,5,6,7-tetrahydro-2H-indazole
1-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
4-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]morpholine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
(1S,5R)-3-benzoyl-N-(2-phenylethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
8-(butan-2-yl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{1-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
1-methyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]azepane-2-carboxamide
4-benzyl-11-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3R,4S)-1-(5-methoxyfuran-2-carbonyl)-4-propylpyrrolidin-3-amine
[3-(2-methoxyethyl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl]methanol
4-amino-2-{4-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
2-(3-chlorophenyl)-1-[3-(pyrrolidin-1-yl)propyl]-1H-imidazole
6-tert-butyl-N-{[1-(methoxymethyl)cyclopropyl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(3-fluorophenyl)-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-one