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N'-cycloheptyl-N-[1-(thiophen-2-yl)propan-2-yl]butanediamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-1H-pyrazole-4-carboxamide
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
3-(3-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-(2-fluorophenoxymethyl)-N-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(1H-indol-2-ylmethyl)-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]pyrrolidin-3-yl]acetamide
(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)({2-[4-(4-fluorophenyl)piperazin-1-yl]-7-methoxyquinolin-3-yl}methyl)amine
1-(3-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propyl)-1H-pyrazole
methyl (2S)-1-(3-{[4-(dimethylamino)phenyl]methyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)pyrrolidine-2-carboxylate
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-(4-ethoxyphenyl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
1-[(4-methylphenyl)amino]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]cyclopentane-1-carboxamide
1-methyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]piperidine-3-carboxamide
3-(4-hydroxyphenyl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}benzamide
N-{[(2S,4S)-4-fluoro-1-[2-(pyridin-4-ylsulfanyl)acetyl]pyrrolidin-2-yl]methyl}propane-1-sulfonamide
N-[2-(4-chlorophenyl)ethyl]-N-(pyridin-4-ylmethyl)oxolane-3-carboxamide
2,3-dimethyl-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
(1S)-1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-methylpiperidine
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
N-(1-{1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
(1R,3S,5S)-8-(7-methoxy-4-methylquinazolin-2-yl)-8-azabicyclo[3.2.1]octan-3-ol
N-(3-fluorophenyl)-6-[2-(2-methoxyphenoxy)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(3,4-dichlorophenyl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
2,6-dimethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidine-4-carboxamide
[(3,5-dichloropyridin-4-yl)methyl]({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(propan-2-yloxy)benzamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidin-2-amine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-cyclopropyl-N-{[3-(difluoromethoxy)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
N-methyl-N-(3-methylbutyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(morpholin-4-yl)-6-(pyrimidin-5-yl)pyrimidin-4-amine
N-{[8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}oxane-4-carboxamide
2-[4-(1H-imidazol-1-yl)benzoyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one
[2-(diethylamino)ethyl]({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})ethylamine
N-(dimethyl-1H-1,2,4-triazol-3-yl)-2-methyl-4-phenylpiperazine-1-carboxamide
1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-4-phenylbutane-1,2-dione
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[4-(furan-2-yl)benzoyl]-3-(2-methoxybenzoyl)piperidine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-2-ylsulfanyl)acetamide
3-(1H-1,3-benzodiazol-2-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2,6-dimethoxypyridine-3-carboxamide
3-[4-(4-hydroxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
N-[(2S)-2,3-dihydroxypropyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)ethyl]-2-phenoxyacetamide