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1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
2-(adamantan-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
2-[4-(dimethylamino)phenyl]-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]ethan-1-one
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(2-methylpropyl)acetamide
2-(3-methylbut-2-en-1-yl)-8-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
6-(cyclobutylamino)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
3-cyclopropyl-5-({5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}methyl)-1-phenyl-1H-1,2,4-triazole
2-(2-chlorophenyl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N,5,7-trimethyl-N-[2-(oxan-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
N-(2-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-3-carboxamide
6-methyl-N-[(6-methylquinolin-5-yl)methyl]-4-oxo-4H-pyran-2-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
(2R,6R)-10-methoxy-4-(1H-pyrrole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(4-{9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}piperidin-1-yl)ethan-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(5-methylfuran-2-yl)methyl]benzamide
ethyl 2-[(2-{[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]carbamoyl}phenyl)amino]acetate
5-chloro-2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidine
N-(2-methoxyethyl)-1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[(5-methylfuran-2-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-[(2-fluoro-5-methoxyphenyl)methyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(2-methoxyphenoxy)-1-(5-methoxypyrimidin-2-yl)piperidine-4-carboxylic acid
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-cyclopropyl-1,2,4-oxadiazole
2-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}quinolin-4-ol
N-[cyclopropyl(4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-(4-methoxyphenyl)-7-(prop-2-en-1-yl)-2-(thiomorpholine-4-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(3R,9aR)-3-methyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(1S,5R)-6-(2-methoxyethyl)-3-(quinolin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-chloro-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-fluorobenzamide
methyl 4-(4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)benzoate
7-(cyclopropylmethyl)-2-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,7-diazaspiro[4.5]decane
2-(3,4-dichlorophenyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]morpholine
3-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-{2-[1-(thiophen-3-ylmethyl)piperidin-2-yl]ethyl}morpholine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-benzyl-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-(2-methylphenyl)-3-[4-(quinazolin-4-yl)piperazin-1-yl]propanamide
6-[(2,6-dimethoxyphenyl)methyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,2-dimethyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}thiomorpholin-3-one
2-{4-[(2,6-difluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
1-[4-(piperidin-3-yl)benzoyl]-4-(pyridin-4-yl)piperazine
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
1-cycloheptyl-6-oxo-N-(prop-2-en-1-yl)piperidine-3-carboxamide
N,N-dimethyl-4-[4-(piperidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]aniline