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3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(4-chlorophenyl)methyl]-8-(2-hydroxy-3-methylbutanoyl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-3-yl}acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-amine
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)propanamide
[1-({1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1H-pyrazol-4-yl)propanamide
1-(1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-3-methylbutan-1-ol
5-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
methyl N-(2-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)carbamate
N-[(3R,4S)-4-cyclopropyl-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-2-methoxyacetamide
2-methyl-5-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}pyridine
3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{3-[4-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)piperidin-1-yl]phenyl}pyridine-3-carboxamide
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
2-methoxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
8-(1-benzothiophen-2-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(4-acetylphenoxymethyl)-N-[(2-methoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
4-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-N-(pyridin-3-yl)benzamide
methyl (2S)-1-{2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}pyrrolidine-2-carboxylate
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-5-phenyl-1,2-oxazole-3-carboxamide
methyl 5-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-ethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-[(2,5-difluorophenyl)methyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
3-methyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyridine
1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]piperidine-1-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyridin-2-amine
N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-2-(4-fluoro-3-methylphenyl)acetic acid
methyl 3-cyclobutaneamido-5-[(pentan-3-yl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-acetyl-N-methyl-N-(oxan-2-ylmethyl)thiophene-3-carboxamide
2-[5-(4-phenyl-1H-imidazol-5-yl)furan-2-yl]benzonitrile
N-[(3R,4S)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole
5-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-[3-(piperidin-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
2-[5-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(4-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl]acetic acid
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
2-(3-fluorophenyl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-N-(thiolan-3-yl)pyridin-2-amine
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
1-(4-fluorophenyl)-N-(furan-3-ylmethyl)cyclopropane-1-carboxamide
(1S,5R)-6-propyl-3-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane