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2-{5-[(2S)-2,3-dihydro-1H-indole-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-1,3-thiazol-4-yl}methanol
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
2-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}acetic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
3-(1,3-benzothiazol-5-yl)-1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}urea
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
8-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-(1-hydroxy-2-methylpropan-2-yl)-N-(pyridin-2-ylmethyl)-1-benzothiophene-2-carboxamide
2-methoxy-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(3,5-dimethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
1-(4-hydroxypiperidin-1-yl)-2-(4-{4-[methyl(2-phenylethyl)amino]piperidin-1-yl}phenyl)ethan-1-one
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
1-(3-fluorophenyl)-6,6-dimethyl-N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(4-methoxyphenyl)-N-[2-methyl-1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)propyl]acetamide
N3-ethyl-N1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}pyrrolidine-1,3-dicarboxamide
6-(azepane-1-carbonyl)-N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
2-(pyridin-4-yl)-4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}quinoline
2-(3,4-dimethoxyphenyl)-1-[3-(pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-methyl-N-(oxan-2-ylmethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
4-(4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-[(3-fluorophenyl)methyl]-4-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperazine
4-chloro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methoxybenzamide
5-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-ethyl-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-propylpiperidin-3-yl}methanol
N-methyl-N-(2-methylpropyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N,N-dimethyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[(2S)-2-amino-2-cyclohexylacetamido]-N-tert-butyl-2-methylbenzamide
2-[4-(2-methoxyphenyl)piperidine-1-carbonyl]-1-methylazepane
8-(2-methyl-1-benzofuran-5-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-(2,2-difluoroethyl)-2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-7-fluoro-4-methylquinoline
4-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
5-(2-fluorophenyl)-N-[3-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-hydroxy-1,2-oxazolidin-2-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
(isoquinolin-5-ylmethyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-(4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-4-oxobutyl)acetamide
1-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}cyclopentan-1-ol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4,4,4-trifluorobutanamide
3-(3-methoxyphenyl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
7-[2-(morpholin-4-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-(1,2-oxazol-3-ylmethyl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
4-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole