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{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-{5-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxymethyl]-1,2,4-oxadiazol-3-yl}pyrazine
N-(2-{1-[(4,5-dichlorothiophen-2-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
N-[2-(oxolan-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)morpholine
(2S,4R)-N,N-diethyl-1-methyl-4-(2-methyl-1-benzofuran-5-amido)pyrrolidine-2-carboxamide
N-({8-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
4-(4-chlorophenyl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}butan-1-one
3-ethyl-5-{[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4,5-dihydro-1,2-oxazole
2-[4-(dimethylamino)phenyl]-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
methyl 1-methoxy-2-oxo-8-(3-phenyl-1H-pyrazole-5-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxypyridin-3-yl)propanamide
methyl[(3-methylpyridin-4-yl)methyl]{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}amine
N-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
4-{2-[benzyl(methyl)carbamoyl]ethyl}-N-butylpiperidine-1-carboxamide
3-(cyclopropylmethyl)-1-(3,3,3-trifluoropropanesulfonyl)piperidine-3-carboxylic acid
1-[2-(2,4,6-trimethylphenyl)pyrimidin-4-yl]piperidin-4-ol
1-[2-methoxy-6-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-4-ethylpiperazine
N-[(5-ethylpyridin-2-yl)methyl]-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-[2-(dimethylamino)ethyl]-8-(3-methoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
1'-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)propanamide
6-methyl-N4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
5-(3-{4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
1-methyl-1'-[2-(4-methylphenoxy)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
(2R,3R)-3-[3-(3-methylphenoxy)azetidin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2E)-3-(1,3-benzothiazol-2-yl)-N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]prop-2-enamide
2-phenoxy-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
5-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]pyridin-2-amine
N-(3-chloro-4-methoxyphenyl)-3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]propanamide
2-{4-cycloheptyl-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-ethyl-5-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-{ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}-2-(4-fluoro-3-methylphenyl)acetic acid
({4-ethyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(pyridin-2-ylmethyl)-1-{1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}piperidine-4-carboxamide
2-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-2,8-diazaspiro[4.5]decane
1-methyl-6-(pyridin-3-yl)-N-[4-(pyrrolidin-1-yl)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}piperidine-1-carbonyl)pyridine
2-(2,4-dichlorophenoxy)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]acetamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide