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4-[2-(4-fluorophenoxy)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-7-fluoro-3-methyl-1H-indole
2-(2-aminoethyl)-N-[2-(4-fluorophenyl)ethyl]quinazolin-4-amine
(2R,3R,6R)-3-(4-fluorophenyl)-5-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclohexyl-3-ethyl-4-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
9-(2-aminopyridine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
4-(2-fluorobenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-ethylpyridine-4-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-4-fluorobenzamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethan-1-one
5-[4-(1H-1,2,4-triazol-1-yl)phenoxy]-1-azabicyclo[3.2.1]octane
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
4-{2-[1-(5-methylthiophene-3-carbonyl)piperidin-2-yl]ethyl}phenol
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
ethyl 4-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}amino)cyclohexane-1-carboxylate
N-cyclopropyl-1-[1-(2-phenoxyethyl)piperidin-4-yl]piperidine-3-carboxamide
5-ethyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
N-[(4-fluorophenyl)methyl]-4-hydroxy-2-methyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[3-(dimethylamino)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{3-[(4-methoxyphenyl)methyl]-5-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl}acetic acid
6-[(diethylamino)methyl]-N-(1-hydroxy-2-methylpropan-2-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(4-fluorophenyl)piperazin-2-one
1-{3-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
2-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-7-(morpholine-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-(2-oxo-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,3-oxazolidin-2-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
4-[(2-chlorophenyl)methyl]-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,4-diazepan-5-one
4-ethyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
1-(3-methoxybenzoyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(thiophene-3-carbonyl)-1,4-diazepan-2-one
N-({1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}methyl)acetamide
N-[(2-chlorophenyl)methyl]-5-[(dimethylamino)methyl]-N-(prop-2-en-1-yl)furan-2-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methylpyridine-3-carboxamide
1-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
5-[(2,3-difluorophenyl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-(4-{2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazin-1-yl)-N,N-dimethylacetamide
2-hydroxy-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(methylsulfanyl)butan-1-one
4-[(2E)-3-phenylprop-2-enoyl]piperazine-2-carboxylic acid
1-cyclopentyl-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
3-{5-[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-4-phenyl-1H-imidazol-1-yl}propanoic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(2-hydroxyethoxy)ethyl]-5-methylpiperidin-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-(1-benzylpiperidin-4-yl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
[2-(3,4-dimethoxyphenyl)ethyl]({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
4-(1H-imidazol-4-ylmethyl)-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(4-{1-[3-(1,3-thiazol-4-yl)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine