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3-{[2-(3-fluorophenyl)azepan-1-yl]methyl}pyridin-2-amine
N-[2-(2-fluorophenyl)ethyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(4-chloro-2-ethylphenyl)-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
(1S,9S)-11-{[6-methyl-4-(thiomorpholin-4-yl)quinazolin-2-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-methoxy-2-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
(4aS,8aR)-1-(3-aminopropyl)-6-(1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N,2-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
6-(2,5-dihydro-1H-pyrrol-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
4-methyl-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}azepan-4-ol
[(3R,4S)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]morpholine
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-amino-7-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-3-methoxypropan-1-one
N-{3-methyl-1-oxo-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]butan-2-yl}acetamide
2-{5-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3-phenyl-1H-1,2,4-triazol-1-yl}acetic acid
1-methyl-3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[1-(pyridin-3-yl)pentyl]urea
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl]propanoic acid
2-methoxy-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)acetamide
1-(2-methoxyacetyl)-N-[(2-phenylphenyl)methyl]piperidine-4-carboxamide
3-[5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
2,5-dimethyl-3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethylbenzamide
1-{1-[6-(3-methoxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
{5-fluoro-7-[4-(pyrrolidin-1-ylmethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}acetamide
5-cyclopropanecarbonyl-1'-(1-methyl-1H-imidazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
1-{4-[(3,5-dichloropyridin-4-yl)methyl]piperazine-2-carbonyl}-4-methylpiperazine
methyl 5-(6-chloropyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(4-chlorophenoxy)-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
4-[2-({4-benzyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)ethyl]morpholine
1-(2-methoxyethyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-butyl-4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-methyl-1,3-benzoxazole-6-carboxamide
N-{1-[({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2H-1,3-benzodioxole-5-carboxamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-methoxy-N-[1-methyl-7-(4-phenylazepane-1-carbonyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazol-5-yl]acetamide
1-ethyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-5-oxopyrrolidine-3-carboxamide
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]propanamide
1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-3-(thiophen-2-yl)propan-1-one