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N-(quinolin-7-yl)-1H-indazole-3-carboxamide
2-{[3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2H-1,2,3,4-tetrazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(7-fluoro-4-methylquinolin-2-yl)piperidin-3-ol
(2R)-2-{4-phenyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}propanamide
(4aR,8aR)-2-[(4-chloro-2-fluorophenyl)methyl]-7-cyclobutanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
1-(2-cyclohexylethyl)-3-hydroxy-3-[({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]piperidin-2-one
4-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-thiazole-5-carboxamide
methyl[(5-methyl-1H-indol-3-yl)methyl]{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
5-(3-fluorophenoxymethyl)-N-methyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-3-carboxamide
5-[(2-chlorophenyl)methyl]-5-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-(2-ethoxyethyl)-2-oxo-1-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-(5-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]imidazolidine-2,4-dione
1-benzyl-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-ethenylphenyl)-3-[1-(methoxymethyl)cyclopentyl]urea
1-{2-[1-(4-fluorophenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(3-chlorophenyl)-N-(2-fluoroethyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(benzyloxy)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
2-(4-chlorophenyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]morpholine
3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole
2-(4-fluoro-3-methylphenyl)-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}acetic acid
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidine
5-(morpholin-4-ylmethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}furan-3-carboxamide
2-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)thiophen-3-amine
(2S,4R)-1-(1H-imidazol-4-ylmethyl)-N-methyl-4-(2-phenoxyacetamido)pyrrolidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}isoquinoline-3-carboxamide
2-cyclohexyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(4aS,8aR)-6-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)-1-(pyrrolidin-1-yl)ethan-1-one
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-N-ethylpyrimidin-2-amine
(4aS,8aR)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-N-[3-(hydroxymethyl)-2-methylphenyl]benzamide
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-1H-indole-6-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
2-(2,6-dimethoxypyrimidin-4-yl)aniline
[(2-cyclohexylpyrimidin-5-yl)methyl](ethyl)(oxan-4-ylmethyl)amine
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(5-{[5-(2-cyanophenyl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydroquinazolin-2-one
1,3,6-trimethyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[(5-chlorothiophen-2-yl)sulfonyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-cyclopropyl-4-methyl-N-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
methyl 4-[4-(2-aminoethyl)-6-oxo-1,6-dihydropyrimidin-2-yl]benzoate
2-[(3,5-difluorophenyl)methyl]-8-(oxan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
methyl 7-oxo-9-(3-phenylpropoxy)-3-(quinolin-7-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2-hydroxypropyl)-9-(pyrrolidine-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methoxy-1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine