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N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-[2-(3-methoxyphenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
8-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-{2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](2-methoxyethyl)(thiophen-2-ylmethyl)amine
N-[2-(dimethylamino)ethyl]-3-{[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]oxy}-N-methylbenzamide
1-(2-methylfuran-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-methyl-5-(1-{[5-(4H-1,2,4-triazol-3-ylsulfanyl)furan-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-(cyclopentylamino)-N-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)benzamide
{2-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-oxoethyl}urea
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[4-(methylsulfanyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-chloro-N-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]benzamide
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,2,6,6-tetramethylpiperidine
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
(2S)-1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
methyl 3-{[3-(2H-1,3-benzodioxol-5-yl)propanamido]methyl}-5-(2-methoxybenzamido)benzoate
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
7-(3-hydroxypyridine-2-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
methyl 2-{methyl[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}acetate
N4-[2-methyl-1-(pyridin-2-yl)propyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
2-[(4aR,7aS)-4-[(5-fluoro-2-methoxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-(4-cyclobutyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(2-fluorophenyl)piperidin-4-ol
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2-methoxyphenyl)methyl]piperazine
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-1-methyl-1H-pyrazole-3-carboxamide
4-{1-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]piperidine-3-carbonyl}morpholine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
4-methoxy-3-[3-(propan-2-yloxy)phenyl]benzamide
1-(3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-oxopropyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]-1-(thiophen-2-ylmethyl)piperidine
4-[1-(2-methylphenyl)-5-[(2-oxopyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]benzamide
methyl 6-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)pyridine-2-carboxylate
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(1-methylcyclohexanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
6-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
N-(1-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2,4-dimethylbenzamide
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-(quinolin-8-ylmethyl)-1,3-oxazole-4-carboxamide
1-(5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
1,3-dimethyl-N-({8-[(2,3,4-trimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-[2-(propylsulfanyl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(pyridin-3-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(4-methyl-1,3-thiazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 4-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-3-yl}piperazine-1-carboxylate
5-amino-N-[3-(2-methoxybenzamido)phenyl]-1H-pyrazole-3-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1-ethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-chloro-2-(methylamino)-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide