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6-(2-aminoethyl)-N-(3-methoxypropyl)-2-methylpyrimidin-4-amine
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
2-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1,3-benzothiazole
N-cyclopropyl-N-({4-[(2,5-dimethoxyphenyl)methoxy]phenyl}methyl)quinoline-2-carboxamide
2-methyl-4-{5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]furan-2-yl}but-3-yn-2-ol
4,6-dimethyl-1-{2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
3-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-[2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-(4-aminopyridine-2-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
(3S,4S)-N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-methoxy-1-(propan-2-yl)pyrrolidin-3-amine
4-{[1-(3-phenylpropyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2,8-dimethyl-N-[3-(pyridin-3-yl)propyl]quinoline-4-carboxamide
5-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-(2-methylpropyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-amine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]-N,N-dimethylaniline
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
3-[3-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1H-indol-1-yl]propanamide
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}spiro[azepane-4,2'-chromene]
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
5-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
4-(hydroxymethyl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]azepan-4-ol
1-ethyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-pyrazole-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
4-(dimethylamino)-N,N-bis(propan-2-yl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
4-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
4-[(2-chlorophenyl)methyl]-1-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-5-one
(2S)-4-methyl-2-[2-(naphthalen-1-yl)-1H-imidazol-1-yl]pentanamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
8-[(4-chloro-2-fluorophenyl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
7-{2,3-dimethyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-2-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(hydroxymethyl)azepan-4-ol
2-(4-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,4-diazepan-1-yl)-1,3-benzothiazole
8-chloro-2-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}quinoline
[(1-{[1-(oxan-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
1,3-dimethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
dimethyl({2-[2-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]ethyl})amine
{1-[(2-phenylpyrimidin-5-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-benzotriazole
2-methyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-phenoxypropanamide
4-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-propoxybenzamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide