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5-[benzyl(methyl)amino]-2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
1-[3-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]-2-(4-methylpiperidin-1-yl)ethan-1-one
N-cyclopropyl-5-[3-(trifluoromethyl)phenoxymethyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
1-[(2-fluorophenyl)methyl]-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
2-cyclopentyl-1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
4-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)phenyl]but-3-yn-1-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(pyrrolidin-1-ylmethyl)benzamide
3-[4-(diphenylmethyl)piperazin-1-yl]-5-phenyl-1,2,4-triazine
[(3R,5R)-5-[(dimethylamino)methyl]-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidin-3-yl]methanol
3-[2-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)propyl]-3,4-dihydroquinazolin-4-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide
3-methyl-3-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1-phenylurea
methyl 2-(azocane-1-sulfonyl)-6-(3-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)acetamide
1-(2-ethoxyethyl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-hydroxypyridine-3-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-(dimethylamino)-N-{3-methyl-1-[7-(3-methylbutanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
5-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
1-(2-methoxy-4-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
(3S,4R)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-benzyl-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2-hydroxyethyl)propanamide
2-methoxy-5-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazol-2-yl}pyrimidine
2-benzyl-9-[3-(methylsulfanyl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(1-cyclopropanecarbonylpiperidin-4-yl)-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
methyl 2-[4-(2-methyl-1,6-naphthyridine-3-carbonyl)-2-oxopiperazin-1-yl]acetate
3-[5-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,2,3-thiadiazole-5-carboxamide
9-[2-(ethylsulfanyl)propanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
1-(furan-2-ylmethyl)-N-propyl-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(3aS,6aS)-2-methyl-5-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1'-(2,4-difluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(2,2-dimethylpropyl)-2-(5-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(1R,7S)-6-(4,4-difluoropiperidine-1-carbonyl)-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-(2-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
[1-(1,7-dimethyl-1H-indole-2-carbonyl)-3-propylpiperidin-3-yl]methanol
(2R)-2-[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
5-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-methoxyphenol
N-(2,2-dimethyloxan-4-yl)-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
2-(4-ethylpiperazin-1-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
3-[5-(2-hydroxypyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-[(2-chlorophenyl)methyl]-1-cycloheptyl-N-methyl-6-oxopiperidine-3-carboxamide
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
4-chloro-N-[(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-3-methylbenzamide