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N-(4-chloro-3-fluorophenyl)-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
2-[(diethylamino)methyl]-4-(6-methoxypyridin-2-yl)phenol
7-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-cyclopropyl-3-{5-[3-(2-fluorophenyl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-(1H-1,3-benzodiazol-1-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanamide
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-methylpiperidine-3-carboxamide
N-[2-(ethylsulfanyl)ethyl]-2-(morpholine-4-carbonyl)pyridin-4-amine
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(2,3-dimethylphenyl)-1H-pyrazole-4-carboxylate
2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-[4-(trifluoromethyl)phenyl]ethan-1-ol
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
5-methanesulfonyl-4-(piperidin-3-yl)-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyrimidine
2-amino-6-(2,6-difluorophenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
3-(2-ethylbutyl)-8-propanoyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(2-phenylethyl)-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
3-cyclohexyl-N-[(3R)-pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
4-{2-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}morpholine
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(2-oxoazepan-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-[2-(furan-2-ylmethoxy)phenyl]thiomorpholine-4-carboxamide
5-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-1-(2-methoxyethyl)piperidin-2-one
N-[1-(3,5-difluorophenyl)cyclopropyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
methyl 3-(2-chlorobenzenesulfonamido)-5-[(3-phenylpropanamido)methyl]benzoate
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N-[2-(dimethylamino)ethyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
5-methoxy-2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
N,N-dimethyl-4-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
4-(cyclopropylmethyl)-1-[2-(4-fluoro-2-methylphenyl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
2-(ethylsulfanyl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)propanamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(piperidin-1-ylmethyl)-1,4-oxazepane
N-[2-(2,4-difluorophenyl)-1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(dimethylamino)-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
9-methoxy-7-(3-methoxyphenyl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]morpholine
4-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
5-(3-oxo-3-{spiro[indene-1,4'-piperidine]-1'-yl}propyl)imidazolidine-2,4-dione
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
2-[4-(4-fluorophenyl)oxane-4-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-(cyclohex-1-en-1-ylmethyl)-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
(3S,4R)-4-(4-fluorophenyl)-1-(4-methoxy-3-methylbenzoyl)pyrrolidine-3-carboxylic acid
3-methyl-7-[(4-phenylphenyl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-methyl-6-(propan-2-yl)-N-[1-(pyridin-2-yl)propyl]pyrimidin-4-amine
1-methyl-2-oxo-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-methyl-8-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,5R)-6-(2,1,3-benzoxadiazol-4-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[4-methoxy-3-({[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)phenyl]acetamide