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N-[4-(1H-indol-2-yl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-(1,2-diphenylethyl)-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidine-2-carboxamide
(5S,9aS,9bS)-2-methyl-5-[2-(naphthalen-1-yl)pyrimidin-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-[3-(dimethylamino)phenyl]acetamide
N-[2-(dimethylamino)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)-2-(thiophen-2-ylformamido)propanamide
6-methyl-4-(4-methyl-1H-imidazol-5-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-{[5-(1-benzothiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-(3-{[({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)carbamoyl]methoxy}phenyl)propanamide
3-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
N-(5-propyl-4H-1,2,4-triazol-3-yl)-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
3-[(3R,4S)-3-[1-(1H-imidazol-1-ylmethyl)cyclopropaneamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
N-{2-[1-(2,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-[3-(1H-imidazol-1-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopropyl-N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
2-methoxy-N-[2-(4-methylmorpholin-2-yl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
N-(4-{[4-(3-cyanopyridin-2-yl)piperazin-1-yl]methyl}phenyl)acetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}propanamide
4-[2-amino-3-cyano-6-(4-hydroxy-3-methoxyphenyl)pyridin-4-yl]benzoic acid
(3aS,6aR)-5-[2-(methylsulfanyl)pyrimidin-4-yl]-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(2,3-dihydro-1H-inden-2-yl)-3-propoxypiperidine
2-[5-(isoquinolin-5-yl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-cyclohexanecarbonyl-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)ethan-1-one
methyl 5-{imidazo[1,2-a]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-[(3,4-dimethoxyphenyl)methyl]-N-[(6-methylpyridin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
N,N-dimethyl-2-[2-(trifluoromethoxy)phenyl]benzamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(3-methylthiophen-2-yl)methyl]benzamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
1,4,6-trimethyl-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydropyridin-2-one
3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-6-methylpyridazine
3-(2-hydroxypropan-2-yl)-N-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}piperidine-1-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
N-[2-(diethylamino)ethyl]-N-ethyl-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]benzamide
2-methoxy-5-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)pyridine