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3-methyl-1-{1-[6-(1,4-oxazepan-4-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
N-(2-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-N-methylmethanesulfonamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-(2-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}quinolin-5-yl)acetamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-[(3-ethoxy-4-methoxyphenyl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-{[(2-chloro-5-sulfamoylphenyl)carbamoyl]amino}cyclopentane-1-carboxamide
1-(2-methoxybenzoyl)-4-[3-(5-methylfuran-2-yl)butyl]piperazine
2-(cyclopropylmethyl)-N-[(4-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-amino-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-4-carboxamide
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-[1-(2-methoxyphenyl)ethyl]-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
methyl 2-{1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-oxopiperazin-2-yl}acetate
1-(oxan-4-ylmethyl)-4-(propan-2-yl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-methyl-N-(2-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)piperidine-3-carboxamide
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-(4-fluoro-2-methoxyphenyl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-fluoro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
2-butoxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-[4-(6-aminopyridin-2-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-indazol-3-yl)acetamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(2-methoxyphenyl)methyl]piperidine-4-carboxamide
4-[3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,4-diazepane-1-carbaldehyde
(1S,5R)-6-[5-(methoxymethyl)furan-2-carbonyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,9S)-11-(4-ethoxypyrimidin-2-yl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(2S,4R)-4-amino-1-[(3,5-dimethoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
3-methoxy-N-[1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
methyl 3-[1-(2-methoxyphenyl)-1H-pyrazole-4-amido]azepane-1-carboxylate
4-[(3,5-dimethoxyphenyl)methyl]-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)methyl]-1λ6-thiane-1,1-dione
N-cyclopentyl-5-(1,2-oxazol-3-yl)-N-{[4-(oxolan-3-yloxy)phenyl]methyl}thiophene-2-sulfonamide
2-methyl-8-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecane
N-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1-(methoxymethyl)-N-methylcyclopropan-1-amine
5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-2-(2-methoxyethyl)pyrimidine
5-{4-[(4-ethoxypiperidin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)-N-(6-methylpyridin-3-yl)benzamide
N-[1-(2-fluorophenyl)piperidin-4-yl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-(propan-2-yloxy)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-{5-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}methanesulfonamide
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]oxolane-2-carboxamide
6-(3-methoxyphenyl)-N-(1-phenylcyclopropyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}acetamide
5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(2-phenylethyl)piperidin-2-one
8-(3-methoxypyrazin-2-yl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(3-methylpyridin-4-yl)methyl]-2-azaspiro[4.5]decan-3-one
N-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(6-methylpyridin-2-yl)piperazine-1-carboxamide