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5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-imidazole-4-carboxylic acid
4-(cyclohex-3-ene-1-carbonyl)-1-cyclohexyl-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-4-(pyrimidin-2-yl)phenoxy]acetamide
2-[3-({[3,3-dimethyl-1-(pyridin-3-yl)butyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
5-(2,5-dimethylfuran-3-yl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1,2,4-triazin-3-amine
5-(4-methoxyphenyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}furan-2-carboxamide
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}acetamide
5-cyclopentanecarbonyl-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(1S,2S)-N2-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2,3-dihydro-1H-indene-1,2-diamine
3-[5-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
4-(1-ethyl-1H-pyrazole-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(2-methylpropyl)piperidine-3-carboxamide
N-benzyl-1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]piperidine-3-carboxamide
(2E)-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}-3-(pyridin-3-yl)prop-2-en-1-one
N-cyclopentyl-2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-methyl-4-[3-methyl-5-(1-methyl-5-phenyl-1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl]piperidine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carboxamide
2-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-6-methyl-4H-pyran-4-one
[(2-fluoro-5-methoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl 4-{4-[(4-cyclopentyl-3-oxopiperazin-1-yl)methyl]-5-methyl-1,3-oxazol-2-yl}benzoate
ethyl 4-[(2-chlorophenyl)methyl]-1-(2-acetamidoacetyl)piperidine-4-carboxylate
3-(2-phenylethyl)-7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
8-[(5-acetylthiophen-3-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-(2-cyclopentylacetamido)-1-methyl-N-(oxan-4-yl)-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-4-chloro-3-methyl-1H-pyrazole-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-{[4-(3-methylphenyl)phenyl]methyl}piperidin-4-yl]pyridine-4-carboxamide
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-ol
(3S,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidine-3-carboxylic acid
N-(1-methyl-1H-1,2,3-triazol-4-yl)-3-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N,6-dimethyl-2-(morpholin-4-yl)pyrimidin-4-amine
(1S,6R)-9-(3-methoxy-5-methylthiophene-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
1-cyclohexyl-4-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-benzyl-N-(quinoxalin-6-yl)-1,3-thiazole-4-carboxamide
1-methyl-4-phenyl-3-[1-(prop-2-ene-1-sulfonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N4-[(1-ethylpyrrolidin-2-yl)methyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
(2S)-2-amino-2-cyclopropyl-N-[1-(4-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
2,5-dimethyl-3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
4-methoxy-2-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(5-methyl-1,2-oxazol-3-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-4-(piperidin-1-ylmethyl)benzamide
3-cyclopropyl-5-(1H-1,2,4-triazol-5-yl)-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
(1S,5R)-6-(2-methoxyethyl)-3-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol