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N-{2-[5-methyl-4-({[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}oxolane-2-carboxamide
(2S)-1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}pyrrolidine-2-carboxamide
4-{4-[3-(3-methylphenyl)piperidin-1-yl]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
1-(pyrrolidin-3-yl)-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperazine
cyclopentyl 4-[(4-acetyl-1,4-diazepane-1-carbonyl)amino]benzoate
3-[(1S,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanoic acid
5-cyclopropyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,3-oxazole-4-carboxamide
N-ethyl-3-(3-hydroxy-3-methylbutyl)-N-[(5-methylfuran-2-yl)methyl]benzamide
[1-(3-{[4-(propan-2-yl)pyrimidin-2-yl]amino}propyl)piperidin-3-yl]methanol
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-2-(4-methoxyphenyl)acetamide
5-{[(1-hydroxycyclohexyl)methyl]amino}-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[1-(thiophen-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[4-(morpholin-4-yl)butyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[4-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(1-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
(2R,6S)-2,6-dimethyl-4-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)morpholine
N-methyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-4-(trifluoromethoxy)benzene-1-sulfonamide
2-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
3-[(3,4-dimethoxyphenyl)methyl]-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[(isoquinolin-5-yloxy)methyl]-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(5-methoxyfuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-{7-[2-(1H-pyrrol-1-yl)acetyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-one
2-(2-acetamidoethyl)-N-[(2-fluorophenyl)methyl]piperidine-1-carboxamide
2-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-(3-methylphenyl)-2-[4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)morpholin-3-yl]acetamide
2-(pyridin-4-ylmethyl)-9-[3-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-6-ethoxyphenol
1-(1-benzofuran-5-carbonyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-chlorophenyl)methyl]-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
3-cyclopropyl-4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
4-tert-butyl-2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenol
(1S,5R)-3-[2-chloro-5-(piperidin-1-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-5-(1H-indol-3-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{4-[2-chloro-4-(cyclopentylcarbamoyl)phenoxy]piperidine-1-carbonyl}pyridin-1-ium-1-olate
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
N-ethyl-6-[methyl(1-methylpyrrolidin-3-yl)amino]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-(3-methylbutyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
2-(1-ethylpiperidin-4-yl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]acetamide
2-[2-(3,3-diphenylpiperidin-1-yl)ethoxy]ethan-1-ol
4-(5-methylpyridin-2-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-ol
3,7-dimethyl-8-{4-[1-(morpholin-4-yl)ethyl]phenyl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
4-(5-fluoro-2-methylphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide