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3-(furan-2-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
methyl (2S,4S,5R)-2-ethyl-4-[ethyl(methyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylate
2-(4-propanoylphenoxy)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
2-amino-7-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-methyl-3-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}methyl)-1,2-dihydroquinolin-2-one
methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-(1-methylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-2-yl)-1H-pyrazole
1-{2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
7-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-methyl-4-[4-({8-methyl-2,8-diazaspiro[5.5]undecan-2-yl}methyl)phenyl]butan-2-ol
4-(7-chloroquinolin-4-yl)-2-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenol
1-[2-(aminomethyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
3-(3-methoxyphenyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
(1S)-3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylpropan-1-ol
N-(4-chloro-3-methylphenyl)-2-{[2-(dimethylsulfamoyl)ethyl]amino}acetamide
3-(3-fluorophenyl)-4-(2-methylquinoline-4-carbonyl)piperazin-2-one
2-methyl-5-propyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-4-amine
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-methylquinoline
ethyl 1-methyl-3-(2-phenoxyethyl)piperidine-3-carboxylate
3-chloro-N-{[8-(pyridine-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[1-(4-methylpyridin-2-yl)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(dimethylamino)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)benzamide
1-(5-methyl-1,2-oxazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
N-[(2R,3R)-1'-cyclohexanecarbonyl-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-[1-(3-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl(oxolan-3-ylmethyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-(4-methyl-6-{[2-(4-methyl-1H-imidazol-2-yl)ethyl]amino}pyrimidin-2-yl)phenol
4-(1H-1,3-benzodiazol-1-yl)-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxylic acid
2-[4-(2,3-dihydro-1,4-benzodioxine-2-amido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
6-fluoro-2-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}methyl)quinolin-4-ol
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
2-{4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4,6-dimethylquinazoline
3-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
6-(benzyloxy)-1-cyclohexyl-4-[2-(1,3-thiazol-4-yl)acetyl]-1,4-diazepan-2-one
N-[2-(diethylamino)ethyl]-5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-4-yl]propanamide
3-({[(dimethyl-1,3-thiazol-2-yl)methyl]amino}methyl)-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-methyl-2-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-(1-methyl-3-oxopiperazin-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
(4aR,7aS)-1-ethyl-4-(3-hydroxypropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N,N-dimethylpyridin-2-amine
2-({[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}methyl)-3,4-dihydroquinazolin-4-one
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-{1-[(3-methoxyphenyl)methyl]-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
N-(1-benzylpiperidin-4-yl)-7-oxo-2-(pyridine-3-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
9-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-N-ethylpyrrolidine-3-carboxamide