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4-[1-(1-benzyl-1H-pyrazole-4-carbonyl)azetidin-3-yl]pyridine
5,7-dimethyl-4-{[2-(trifluoromethyl)morpholin-4-yl]sulfonyl}-2,1,3-benzoxadiazole
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[(2E)-3-phenylprop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
5-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)pyrimidin-2-amine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-(dimethylamino)pyridine-3-carboxamide
1-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
1-(2-methoxyethyl)-4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-2-one
2-cyclopentyl-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-4-methylpyrimidin-2-amine
N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(oxolane-2-carbonyl)-4-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-(2-fluorophenyl)-1-methyl-3-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
(3R,5R)-N-[2-(3,4-dimethylphenoxy)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
methyl 4-(2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)butanoate
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[3-(1H-pyrazol-1-yl)propyl]pyridin-2-amine
(2S,4R)-4-amino-1-[2-(2,4-dimethoxyphenyl)acetyl]-N-ethylpyrrolidine-2-carboxamide
(3aR,6aR)-2-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1-[(1-ethyl-1H-indol-5-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
N-[1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-phenoxyacetamide
3-(3-hydroxy-3-methylbutyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2,3-difluoro-N-methylbenzamide
1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]isoquinoline
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(3-ethoxybenzoyl)piperidine
N-[3-(3-methoxyphenyl)phenyl]-1-(1H-pyrazole-4-carbonyl)piperidine-4-carboxamide
4-(4-fluorophenyl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)-1,2,3,6-tetrahydropyridine
2,3-dimethyl-7-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}-1H-indole
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2,6-dimethoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,8aR)-1-(2-aminoethyl)-6-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-(4-methylphenyl)piperidin-4-amine
6-chloro-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-methylimidazo[1,2-a]pyridine-3-carboxamide
4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]quinolin-2-amine
1-(4-fluorophenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}cyclopropane-1-carboxamide
4-[1-benzyl-5-(2-cyclopentylacetyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
3,5-dimethoxy-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)benzamide
1-(diphenylmethyl)-N-(quinolin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(2,2-diphenylethyl)-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N'-(2-methylphenyl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanediamide
3-(azepane-1-carbonyl)-1-ethyl-N-[(3-fluoro-4-methylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2-hydroxyethyl)-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-butyl-N-methylacetamide
5-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
2-(4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
N,4-dimethyl-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
N-[1-(4-{[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]carbamoyl}phenyl)-1H-pyrazol-4-yl]-2,4-dimethylbenzamide
5-cyclopropyl-N-[2-(2-hydroxyethoxy)ethyl]-3-methyl-1H-pyrazole-4-carboxamide