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methyl (2S)-2-{[5-(3,4-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylbutanoate
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
(3S,4R)-4-(2-methylphenyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}pyrrolidine-3-carboxylic acid
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
5-[4-(5-methyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
5-(3-methoxyphenyl)-3-[4-(2-methoxyphenyl)piperazin-1-yl]-1,2,4-triazine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-8-fluoro-N-methylquinoline-2-carboxamide
4-{2-[(4-chlorophenyl)methyl]benzoyl}morpholine
N-(3-{4-[(2-cyclopentylacetamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-3-(pyridin-3-yl)propanamide
4-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-4-yl}-5-methylpyrimidine
1-methyl-4-[4-(2-phenylethyl)piperidine-1-carbonyl]imidazolidin-2-one
(3R,4R)-1-[(8-methoxyquinolin-2-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
4-benzyl-N-(4-chlorophenyl)-4-(hydroxymethyl)piperidine-1-carboxamide
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-[methyl(pyridin-2-ylmethyl)amino]acetamide
3-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-1-[2-(trifluoromethoxy)phenyl]urea
1-(4-phenyl-1H-imidazole-5-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
5-methanesulfonyl-4-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]-2-methylpyrimidine
N-[(5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
5-chloro-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-phenyl-1H-indole-2-carboxamide
2-[4-(naphthalen-1-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
8-[4-(ethylamino)pyrimidin-2-yl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-(cyclohexylmethyl)-N-methyl-4-(pyridin-2-ylsulfanyl)-N-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethyl-1,2-dihydropyridin-2-one
2-ethoxy-1-{4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-methyl-6-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)pyrimidin-4-ol
N-[(5-chlorothiophen-2-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
4-{3-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
1-methyl-8-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(1,2,3,4-tetrahydroisoquinolin-5-yl)thiophene-2-carboxylic acid
1-[2-(cyclohexylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
8-(2-aminoacetyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[(2-fluorophenyl)methyl]piperazine
N-ethyl-N-[(2-fluorophenyl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-(3-butoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine
1'-(3-methylfuran-2-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{4-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]thiophen-2-yl}ethan-1-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
5-tert-butyl-4-({3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}methyl)furan-2-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[3-(pyrrolidin-1-yl)butyl]amine
N-[3-(4-methylpiperazin-1-yl)propyl]-3-(1H-pyrazol-4-yl)benzamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(cyclopropylmethyl)piperidine-3-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(cyclohex-1-en-1-yl)acetamide
N-(5-hydroxyadamantan-2-yl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
(2S)-2-amino-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]butanamide
1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
N-[(3R,4S)-1-methanesulfonyl-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide