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1-(4-benzoylpiperazin-1-yl)-2-(prop-2-en-1-ylsulfanyl)ethan-1-one
2-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-(2-oxo-1,3-oxazolidin-3-yl)-N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
1-(2-methoxyethyl)-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-(propan-2-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-4-carboxamide
1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-4-methoxypiperidine
2-{[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]methyl}-6-fluoroquinolin-4-ol
1-[3-(4H-1,2,4-triazol-4-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
3-{[(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-1,2,4-triazol-3-amine
N-[3-(4-{[2-(2-chlorophenoxy)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2,5-dimethylfuran-3-carboxamide
2-[(2-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
5-(4-fluorophenyl)-N-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1,2,4-triazin-3-amine
1-[(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
5-[4-(1H-imidazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydroisoquinoline
2-[4-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)phenyl]pyridine
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
5-(2-cyclopentylacetamido)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-(4-{4-[(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
2-methyl-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyrimidine
N-{2-[ethyl(methyl)amino]-2-methylpropyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]propan-1-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(2-fluorophenyl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
N-[(2R,3R)-1'-(3,4-dimethylbenzoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-6-methyl-2-propylpyrimidin-4-amine
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-(pyrrolidine-1-carbonyl)pyridine
5-[2-(benzylamino)ethyl]-1-[(2-methylphenyl)methyl]pyrrolidin-2-one
[(3R,5R)-1-[2-(methylsulfanyl)benzoyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
5-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}[2-(1H-1,2,4-triazol-1-yl)propyl]amine
(4aS,7aR)-1-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(but-2-yn-1-yl)-5-[1-(naphthalene-2-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[1-(3-methoxy-5-methylthiophene-2-carbonyl)piperidin-4-yl]piperidin-4-ol
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
(1S,4S)-5-[(2R)-3-hydroxy-2-methylpropyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-({1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
N-[2-(2-chloro-6-methylphenoxy)ethyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-(3-cyanopyridin-2-yl)-N-(1-cyclopentyl-1H-pyrazol-5-yl)piperazine-1-carboxamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(2-phenoxyethyl)piperazine
N-({8-[(4-ethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methylpropanamide
3-cyclopropyl-N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-5-carboxamide
[1-(ethylsulfanyl)propan-2-yl]({[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl})amine
3-(4-methoxy-2-methylbenzoyl)-1-(2,2,2-trifluoroethanesulfonyl)piperidine
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[(3-fluorophenyl)methyl]piperazine
[1-(3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]methanol
(2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[(oxan-4-yl)carbamoyl]pyrrolidine-2-carboxylic acid
1-methyl-4-{[(2R,5S)-5-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}oxolan-2-yl]methyl}piperazine