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2-methyl-8-{[4-(5-methylfuran-2-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
methyl (2S)-2-[(4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}phenyl)formamido]-3-methylbutanoate
2-amino-4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidine-5-carboxamide
6-(cyclopropylmethoxy)-4-(2,3-dimethylquinoxaline-6-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)({[5-(methoxymethyl)furan-2-yl]methyl})methylamine
ethyl 1-[(4-methoxyphenyl)methyl]-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{2-oxo-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(butan-2-yl)-1,3-oxazole-4-carboxamide
8-[(2S)-2-aminohexanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-4-yl)piperazine
methyl 3-cyclohexaneamido-6-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
3-[1-(thiolan-3-yl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
{3-[(2-fluorophenyl)methyl]-1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}methanol
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-N-(3-hydroxypropyl)piperidine-3-carboxamide
2-methyl-4-(4-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
4-[3-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)propanamido]benzamide
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1-[(4-methylphenyl)methyl]-1H-1,3-benzodiazole
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
methyl 3-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(5S,9aS,9bS)-5-(3-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-{1-[(3-propoxyphenyl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
3-(diphenylmethyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(3-fluorophenyl)methyl]-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
2-(cyclopropylmethyl)-9-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
7,8-dimethyl-4-(3-methylpiperidine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
1-(4-chloro-2-methoxybenzoyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
(1R,2R,6S,7S)-4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(1-benzofuran-2-ylmethyl)-4-(1H-imidazol-1-ylmethyl)piperidine
6-[(3-hydroxy-3-phenylpyrrolidin-1-yl)methyl]pyridine-2-carboxylic acid
3-[(2-aminopyrimidin-5-yl)methyl]-3-methyl-1-[2-(propylsulfanyl)phenyl]urea
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-[3-oxo-3-(pyrrolidin-1-yl)propyl]pyrrolidin-2-one
3-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3,9-diazaspiro[5.6]dodecan-10-one
2-(4-fluorophenyl)-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]acetamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-6-methoxypyrimidine
N-[(7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(thiophen-2-yl)acetamide
1-[2-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-(2-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
methyl 1-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxylate
1-cyclohexyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
4-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-{2-[5-methyl-4-({[4-(2-methylpropyl)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}oxolane-2-carboxamide
1-({4-[(2,3-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
3-{[1-(dimethylcarbamoyl)ethyl](methyl)sulfamoyl}-N-(2-fluoroethyl)benzamide
N-methyl-1-[2-(piperidin-1-yl)ethyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-chloro-N-(2-methoxyethyl)-4-({1-[(methylcarbamoyl)methyl]piperidin-4-yl}oxy)benzamide
1-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(thiophen-2-ylmethyl)urea
ethyl 1-[2-(methylsulfanyl)acetyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-(3-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one