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N-[2-methyl-2-(morpholin-4-yl)propyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(cyclohex-1-en-1-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
(3aS,6aS)-2-(cyclopropylmethyl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(2S)-2-aminopentanoyl]-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[6-(4-methoxyphenyl)pyridine-3-carbonyl]-4-phenylazepane
12-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonane-7-carbonyl}-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
N-(2-methanesulfonylethyl)-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
14-(3-hydroxy-4-methoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N,N,4-trimethyl-3-{[methyl(2-methylprop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]propanamide
(1S,5R)-6-(5-fluoropyridine-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(methylamino)pyridine-4-carboxamide
methyl[2-methyl-2-(morpholin-4-yl)propyl]{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
6-{[(1R,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1-methyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
3-(3-{6-[(3-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
4-(1H-imidazol-2-yl)-1-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-1,2,3-triazole
3-[5-(2-phenylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-(1,4-dioxan-2-ylmethyl)-N,3,6,7-tetramethyl-1-benzofuran-2-carboxamide
N-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-{[7-(2,4-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-fluorobenzamide
4-hydroxy-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-(furan-2-ylmethyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
3-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
9-(4-hydroxybenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
2-{1-cyclopentyl-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(1S,5R)-3-[2-(4-methoxyphenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methoxyethyl)-8-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(pyridin-4-yl)propan-1-one
N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-3-(5-phenylpentanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2-phenoxyethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-{1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-2-methyl-1,4-oxazepane
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-[(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
5,5-dimethyl-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-oxazolidine-2,4-dione
4-[(3-chlorophenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[5-(2-chloro-4-fluorophenyl)-1H-1,3-benzodiazol-2-yl]methanol
1-[4-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(pyridine-2-carbonyl)piperidin-3-yl]propanamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(pyridin-2-yl)ethan-1-one
1-[1-(2-phenylethyl)piperidin-4-yl]-N-[(1s,4s)-4-aminocyclohexyl]piperidine-3-carboxamide
methyl 1-[(3R,5S)-5-(azepane-1-carbonyl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(2-methylpropyl)-2-(oxan-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[(3-methoxyphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}-4-(3,3,3-trifluoropropyl)pyrimidine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)(2-phenylethyl)amine