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4-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
6-(azocane-1-carbonyl)-5-methyl-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
1-ethyl-4-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(2E)-3-(3-fluorophenyl)-1-{4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}prop-2-en-1-one
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
5-methoxy-2-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H-pyran-4-one
1-{1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-cycloheptyl-6-oxo-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-{3-[(3-methoxypyrrolidin-1-yl)sulfonyl]benzoyl}-N-methylpiperidin-4-amine
3-(2-chlorophenyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(3-hydroxyphenyl)propanamide
N-{1-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
ethyl 3-(3-phenylpropyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-3-carboxylate
1-[(2-methoxyphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazine
N-(2,5-dihydroxy-2-methylpentyl)-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
(1S,5R)-6-(2-methoxyethyl)-3-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(2-fluorophenyl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methoxybenzamide
N3,N5-dimethyl-1-(3-methylbutyl)-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-{5-[2-chloro-5-(piperidin-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
2-amino-7-(1H-indazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
4-(4-methyl-1H-pyrazol-1-yl)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
N-(2-methylbutyl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N,6-dimethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-benzyl-4-({4-[2-(methoxymethyl)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
4-[4-(3-fluorophenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
methyl(pyrrolidin-3-ylmethyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-(4,4,4-trifluorobutanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(furan-2-ylmethyl)-5-[1-(2-phenoxypropanoyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-cyclohexyl-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-[6-(3-methoxyphenoxy)pyridin-3-yl]-3-propoxypiperidine-1-carboxamide
N,1,3-trimethyl-N-{2-phenyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]ethyl}-1H-pyrazole-5-carboxamide
({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amine
1-{2-[4-(hydroxymethyl)phenyl]acetyl}-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(furan-3-carbonyl)-1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3,3,5,5-tetramethyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}cyclohexan-1-amine
(2S)-1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidine-2-carboxamide
(4-{[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}oxan-4-yl)methanol
1-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
methyl 2-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carboxylate
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]benzamide
1-{2-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-cyclopropyl-1-({1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)-1H-1,3-benzodiazole
(3aR,6aR)-2-methanesulfonyl-5-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-hydroxybutyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide