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1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-benzoyl-N-[3-(3-chlorophenyl)phenyl]piperidine-4-carboxamide
N-(1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
(3R,4S)-4-cyclopropyl-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidin-3-amine
1-methyl-5-(2-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)-1H-1,2,4-triazole
1-(4-methyl-1,3-thiazol-2-yl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
6-[({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]pyrimidin-4-ol
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-amino-4-[4-(2-hydroxyethoxy)phenyl]-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-acetyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
(3R,4R)-4-cyclopropyl-1-[1-(2-methoxyphenyl)piperidin-4-yl]-3-methylpiperidin-4-ol
2-(2-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
1-(furan-3-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-butyl-8-{thieno[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
(1R,5R)-6-[(2-fluoro-4-methoxyphenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperidin-2-yl}methanol
N-[(3,4-dimethoxyphenyl)methyl]-4-oxo-N-(pyridin-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-(prop-2-en-1-yl)urea
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-4-methyl-2-phenylpyrimidine-5-carboxamide
1,4,6-trimethyl-3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
N6-benzyl-N5-methyl-N5-[2-(pyridin-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(3,4-dimethoxyphenyl)-4-{4-[2-(thiophen-2-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1-benzofuran-4-one
{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}(4,4,4-trifluorobutan-2-yl)amine
3-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-benzyl-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(cyclohexylmethyl)-N3-ethyl-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-(3-methoxyphenoxymethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(2,3-dimethoxyphenyl)-1H-imidazole
1-(3-phenylpropyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-methyl-6-[(1,2,3,4-tetrahydronaphthalen-2-yl)amino]heptan-2-ol
5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidin-2-amine
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(piperidine-1-carbonyl)pyrazine
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-3-(pyrrolidin-1-yl)propan-1-one
3-(4-fluoro-2-methoxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methylphenyl)acetamide
N-(2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
1-(pyrimidin-2-yl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
4-(propylsulfamoyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amine
2-(2-{[2-(dimethylamino)ethyl]carbamoyl}ethyl)-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbutyl)piperidine
2-methyl-2-(pyrrolidin-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-[4-(benzenesulfonyl)piperazin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
(1S,5R)-3-[2-(2-ethoxyethoxy)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(pyridin-3-yl)-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
6-(2,5-dimethylphenyl)-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1r,4r)-4-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}cyclohexan-1-ol