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[(diphenyl-1H-1,2,4-triazol-5-yl)methyl](methyl)(pyridin-3-ylmethyl)amine
9-methoxy-3-{2-[4-(methylsulfanyl)phenyl]acetyl}-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
4-[(2-aminopyridin-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2,5-dioxo-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide
4-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
1-ethyl-3-(propan-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
benzyl[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
3-(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-1,2,3-triazol-1-yl)propane-1,2-diol
1-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1H-imidazole-4-sulfonamide
N-[1-(pyridin-4-yl)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
7-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-fluoro-5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(1S,4S)-2-[5-(naphthalen-1-yl)-1,2,4-triazin-3-yl]-2-azabicyclo[2.2.1]heptane
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-methylpropanamide
2-{[4-(4-acetylphenyl)-5-(2,2-dimethylcyclopropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]thiophene-3-carboxamide
N-[3-({[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3-dimethylbenzamide
(2E)-N-({3-methyl-7-[2-(morpholin-4-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
1-(4,6-dimethylquinazolin-2-yl)-N-[(2-methylphenyl)methyl]piperidin-4-amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-ethyl-N-methylpyrimidin-2-amine
5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-methylphenyl)(pyridin-4-yl)methyl]propanamide
1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)ethan-1-one
5,6-dimethyl-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(4-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
6-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-(2-chlorophenyl)-3-(2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1-methylpyrrolidine-2,5-dione
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(naphthalen-1-ylmethyl)acetamide
3-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-[2-(2-fluorophenyl)-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
1-(2-methylpropyl)-4-{1-[1-(trifluoromethyl)cyclopropanecarbonyl]pyrrolidin-3-yl}piperidine
2-[(2-amino-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)amino]ethan-1-ol
dimethyl[2-(4-{[4-(methylsulfanyl)phenyl]methyl}morpholin-2-yl)ethyl]amine
2-{4-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]morpholin-3-yl}-N-(3-fluoro-2-methylphenyl)acetamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-ethyl-4-methyl-1,3-oxazole
3-amino-1-[(2-butyl-1H-imidazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyridin-3-yl)ethyl]acetamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(piperidin-1-yl)acetamide
1-[1-(but-3-en-1-yl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
N-[2-(1-{6-[benzyl(methyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperidin-4-yl)ethyl]acetamide
(3S,5R)-N3-butyl-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
6-[(diethylamino)methyl]-N-[2-(pyrazin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
9-(5,6-dimethylpyrimidin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
5-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione