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N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
4-({3-[3-(trifluoromethyl)phenoxy]phenyl}methyl)-1,4-oxazepan-6-ol
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-methyl-N-(2-methylpropyl)piperidine-3-carboxamide
N-[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-propylpyrrolidin-3-yl]thiophene-3-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-3-yl}methanol
3-{[bis(prop-2-en-1-yl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
9-[(2-methylpyrimidin-5-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(4-phenylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
N-[(2-chloro-4-fluorophenyl)methyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
(4aS,8aR)-6-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-benzyl-8-(dimethyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecane
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
8-methyl-2-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decane
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-3-methylpiperidine
(2S)-2-hydroxy-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
2-(1-benzyl-4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
2-ethyl-9-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-hydroxyazepan-4-yl)methyl]-5-(pyridin-2-yl)thiophene-2-sulfonamide
ethyl 4-[(2-methoxy-5-phenylphenyl)carbamoyl]piperazine-1-carboxylate
N-[(4-chlorophenyl)methyl]-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-(2-hydroxyethyl)-5-(1H-indazole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-methyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
2-(morpholin-4-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{5-[(3-methoxyphenyl)carbamoyl]furan-2-yl}-1H-imidazole-4-carboxylic acid
ethyl 1-[2-(4-chlorophenoxy)acetyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methoxyphenyl)ethyl]acetamide
(2S,4S)-4-(5-chloro-2-hydroxybenzamido)-N-ethyl-1-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-(1-butyl-3-methyl-1H-pyrazol-5-yl)-4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carboxamide
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
[(8-methoxyquinolin-2-yl)methyl](methyl)(quinolin-5-ylmethyl)amine
N-[2-(4-chlorophenyl)ethyl]-2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]acetamide
2,6,6-trimethyl-1-(2-methylpropyl)-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(2-methoxynaphthalen-1-yl)ethyl]-1-methylpiperidine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
3-methyl-5-{2-oxo-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1-(2-hydroxyethyl)-5-(4-methoxyquinolin-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-ethyl-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
2-(4-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenoxy)acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-ethylpyridin-2-yl)methyl]acetamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[(6-methylpyridin-2-yl)methyl]pyridin-2-amine
2-{3-[hydroxy(phenyl)methyl]-5-{imidazo[1,2-a]pyridin-2-yl}-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(cyclohexylmethyl)-4-(3-methyl-1H-pyrazole-4-carbonyl)morpholine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one