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1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine
[2,2-dimethyl-3-(morpholin-4-yl)propyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
(3S,5R)-N3-[2-(dimethylamino)ethyl]-N5-(4-fluorophenyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
8-(2-methyl-1H-pyrrole-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(3aR,7aS)-2-(2-phenoxyethanesulfonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
ethyl 4-[(8R,9aS)-8-hydroxy-1,4-dioxo-octahydro-1H-pyrido[1,2-a]piperazin-2-yl]piperidine-1-carboxylate
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]morpholine
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one
3-{2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
4-{[5-(3-cyclohexyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrimidine
N-methyl-6-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-4-yl)propanamide
3-[(tert-butylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
5-methyl-N4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrrolidine-2-carboxamide
2-butyl-8-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-cyclohexyl-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)acetamide
N-[2-(2,4-difluorophenyl)-1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylthiophene-2-carboxamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(oxolan-3-yl)propanamide
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridin-2-amine
N-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]methanesulfonamide
{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
5-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
(3aR,6aR)-2-acetyl-5-[(5-chloro-2-hydroxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,7-diazaspiro[4.5]decane
1-ethyl-4-{[2-methyl-4-(3-methylphenyl)-5-oxopiperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
4-[2-(dimethylamino)-2-(4-methylphenyl)acetamido]butanoic acid
4-[2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine-4-carbonyl]morpholine
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
(3S,5S)-N-[(2,5-difluorophenyl)methyl]-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
(4aS,8aR)-6-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-imidazol-1-yl)ethyl]-N-methylbenzamide
methyl (2S,4R)-1-[(2-methylphenyl)methyl]-4-(4-phenylbenzamido)pyrrolidine-2-carboxylate
2-methyl-6-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-2,3-dihydropyridazin-3-one
(4aR,7aS)-1-(pyridin-3-ylmethyl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}urea
4-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
[4-(oxan-2-ylmethyl)-1-(3-phenylpropyl)piperidin-4-yl]methanol
1-(2-methoxyethyl)-N-[3-(2-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
N-[(2,6-dimethoxyphenyl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridin-2-amine
2,6-dimethyl-5-{2-[2-(4-methylpentyl)morpholin-4-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl](1,4-dioxan-2-ylmethyl)methylamine
(1R,7S)-3-(2-methoxyethyl)-N-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(2-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methylphenyl)-1,3-oxazolidin-2-one
8-[2-(3-fluorophenoxy)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one