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N-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-methoxybenzamide
2-methoxyethyl N-{[(2S,4S)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}carbamate
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}cyclopentanamine
(3aS,6aS)-5-{[4-(benzyloxy)-2-methoxyphenyl]methyl}-octahydropyrrolo[3,4-b]pyrrole
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-4-(trifluoromethoxy)benzene-1-sulfonamide
2-ethoxy-6-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
N-[(2,3-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
5-(2,4-difluorophenoxymethyl)-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-methyl-4-(1H-pyrazol-3-yl)-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}benzamide
1-(3-chlorophenyl)-4-(4-methoxy-2-methylbenzoyl)-5-methylpiperazin-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-[(2-fluorophenyl)methyl]acetamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}acetamide
3-(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)propanamide
(2S,4R)-4-{[(3-chlorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
4-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-1-carbonyl)pyrimidine
N-[(2R,3R)-1'-(2,3-dimethylbenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
N-cyclopentyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-(4-fluorophenyl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
[2-(2-chlorophenyl)ethyl]({[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-[(1-phenylpyrrolidin-3-yl)methyl]urea
1-[7,8-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
1-(2-methoxyacetyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1-ethyl-1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[5-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
1-(2,4-difluorobenzoyl)-4-[(3-methylphenyl)methyl]-1,4-diazepan-5-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(1,1,3-trioxo-2,3-dihydro-1λ6,2-benzothiazol-2-yl)propanamide
4-[6-(1-hydroxyethyl)pyridin-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one
(4-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
N-methyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
5-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
1-{5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carbonyl}-N,N-dimethylpyrrolidin-3-amine
1-{5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
N5-methyl-N5-[2-(morpholin-4-yl)ethyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-(diphenylmethyl)-5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
1-(2-cyclohexylethyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2,3-difluorophenyl)methyl]-3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
(2S,4R)-N,1-bis(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
8-(4,6-dimethylpyrimidin-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[1-(4-fluorobenzoyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
N-({7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]quinoxaline-5-carboxamide
6-oxo-1-(pyridin-2-ylmethyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
4-{2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carbonyl}piperazin-2-one
7-(3,6-dimethylpyrazin-2-yl)-4-(oxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-methoxy-N-{2-[2-(pyridin-2-yl)ethyl]phenyl}pyrrolidine-1-carboxamide