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2-(6-methoxypyridin-2-yl)-N,N-bis(propan-2-yl)benzamide
2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-6-(2-methoxyphenyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyridine-3-carboxamide
2-(3-phenylpropyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1,3-benzoxazole-5-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-[2-(methylamino)pyrimidine-5-carbonyl]-4-(pyridin-4-yl)-1,4-diazepan-6-ol
2-[1-(2,2-dimethylpropyl)-4-[(6-fluoroquinolin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-{1-[4-(4-methoxyphenyl)-3,3-dimethyl-5-oxopiperazin-1-yl]-3-methyl-1-oxobutan-2-yl}acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethyl-1,3-thiazole-4-carboxamide
4-[2-(4-fluorophenoxy)ethyl]-1-[(1-methyl-1H-indol-3-yl)methyl]-1,4-diazepan-5-one
1-(4-{4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)-2-propylpentan-1-one
1-(7-methoxy-4-methylquinazolin-2-yl)-N-(oxan-4-ylmethyl)piperidine-3-carboxamide
2-[(4aS,7aR)-4-(morpholine-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
methyl (2S,3S)-2-{[1-(4,7-dimethylquinazolin-2-yl)piperidin-3-yl]formamido}-3-methylpentanoate
4-[2-(2-fluorophenyl)ethyl]-3-(pyridin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,3-thiazol-2-amine
4-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]azetidin-3-yl}morpholine
4-[4-(benzyloxy)piperidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
6-methyl-3-[2-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(1-methyl-1H-indazol-3-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[4-(4-methylpiperazin-1-yl)benzoyl]pyrrolidin-3-yl]methanol
(2R,3R,6R)-3-(4-methoxyphenyl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(1H-indole-2-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[4-(diethylamino)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
(2-{2-[1-(2-chlorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-cyclopropyl-4-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
(1R,7S)-3-[4-(propan-2-yl)phenyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(3-phenylpropyl)-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]piperidin-2-one
1-benzyl-8-(2-methylbutyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-5-methoxy-4H-pyran-4-one
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(cyclohexylmethyl)-N3-cyclopropyl-N5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4S)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperidine-3,4-diol
N-[2-(1H-imidazol-4-yl)ethyl]-2-propylpyridine-4-carboxamide
1-(propan-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-4-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-ol
N-[1-(4-fluorophenyl)propyl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
N-cyclopropyl-1-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-(morpholin-4-yl)-2-(pyridin-3-yl)-1-(pyrrolidin-1-yl)ethan-1-one
N,N-dimethyl-5-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)pyridin-2-amine
methyl 3-cyclobutaneamido-5-[(2-methylpropyl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[1-(adamantan-1-yl)piperidin-4-yl]-N-(1-benzylpyrrolidin-3-yl)propanamide
9-benzyl-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(benzyloxy)-8-[3-(3,5-dimethylphenyl)propanoyl]-1,8-diazaspiro[4.5]decan-2-one
1-[(3-fluorophenyl)methyl]-4-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3,5-dimethoxyphenyl)methyl]-4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
1-(4-{2-methoxy-5-[(2S)-4-methyl-2-(propan-2-yl)piperazine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one