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1-(5-phenoxyfuran-2-carbonyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-(3-methylbutyl)pyrrolidin-2-one
(4aR,8aS)-6-(2H-1,3-benzodioxole-5-carbonyl)-1-[2-(3-fluorophenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-benzyl-N-methyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]pyridine-4-carboxamide
2-(2,3-dihydro-1H-inden-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-benzoyl-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[3-(1-propyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}morpholine
methyl (1R,5S,6R)-6-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
5-(2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-1H-1,2,3,4-tetrazole
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
5-[({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine
1-[5-(2-methoxypropan-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
methyl N-(1-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-1-oxopropan-2-yl)carbamate
4-cyclopentyl-N-(5-acetamido-2-fluorophenyl)-1,4-diazepane-1-carboxamide
7-(1-methanesulfonylpyrrolidine-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[4-(4-ethylpiperazine-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
methyl 3-benzamido-5-(cyclohexylamino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
ethyl 4-[1-(3-methoxypropyl)-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
3-({2-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
5-{[benzyl(methyl)amino]methyl}-N-[(3-chlorophenyl)methyl]-1,2-oxazole-3-carboxamide
6-methyl-2-{2-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
3-{1-[4-(1-acetamidoethyl)phenyl]-3,5-dimethyl-1H-pyrazol-4-yl}propanoic acid
5-butyl-1-(3-phenylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
(4aS,8aR)-6-(2,1,3-benzoxadiazole-5-carbonyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
3-{2-[4-cyclohexyl-3-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
1-[3-(1H-imidazol-5-yl)phenyl]-3-[(1-methanesulfonylpiperidin-3-yl)methyl]urea
8-(2-methyl-1,3-thiazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(dimethylamino)propyl]-N-(furan-2-ylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]-N-(pyrimidin-4-ylmethyl)benzamide
1-methyl-4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine-2-carboxylic acid
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]ethan-1-one
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
1-(prop-2-en-1-yl)-2-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
2-[1-butyl-5-(1-cyclopropanecarbonylpiperidin-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
N,N-dimethyl-2-[(1S,5R)-6-[4-(propan-2-yloxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}benzamide
2-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
2-methyl-4-[4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)phenyl]but-3-yn-2-ol
1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-4-(pyridin-4-yl)piperazine