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N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[3-(pyrrolidin-1-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(5-ethylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{4-[1-(1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazol-4-yl]phenyl}acetamide
1'-(6-cyclopropylpyrimidin-4-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{3-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-oxopropyl}-4-fluorobenzamide
N-{3-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-3-oxopropyl}acetamide
2-[(1-ethyl-1H-indol-3-yl)sulfanyl]-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
1-cyclopentyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-6-oxopiperidine-3-carboxamide
6-methyl-5-{5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(2-methylpropyl)-1-(5-methylthiophene-2-carbonyl)-1,4-diazepan-5-one
2-({methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)benzoic acid
(1R,3S)-3-(2-aminoethoxy)-7-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-7-azaspiro[3.5]nonan-1-ol
3-[1-(2-methylpyrimidin-4-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-1-{1'-[(2R)-pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
[1-(5-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxypyridine-2-carboxamide
2-methyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-methyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[1-(2,2,2-trifluoroethyl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-3-yl]pyridine
3-{methyl[4-(pyridin-3-yl)pyrimidin-2-yl]amino}-1-phenylpropan-1-ol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
2-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}azepan-4-amine
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(5-methyl-1H-pyrazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[1-(3-methoxypropyl)-1H-imidazol-2-yl]-2,1,3-benzoxadiazole
4-(5-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-methyl-1H-1,3-benzodiazole
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-methoxyphenyl)piperidine
N,3-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-benzothiophene-2-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,1-dimethyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}pyridine-3-carboxamide
2,5-dioxo-6-(3-propoxypropyl)-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}){[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-{1-[4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)carbamoyl)phenyl]-1H-pyrazol-4-yl}furan-3-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(5-oxopyrrolidin-2-yl)acetamide
2-(dimethylamino)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-phenylethyl)piperidine
N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)cyclohexanecarboxamide
2-methyl-4-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
{2-[(4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}urea
(1S,6R)-9-{5-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
4-(4-{[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
2-chloro-6-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyridine-4-carboxamide
ethyl 2-{[3-(2-{[(3-methoxyphenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]amino}acetate
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-4-yl)propan-1-one
1-(1,2-oxazol-3-ylmethyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide