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N-butyl-N-methyl-3-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
4-({2-[1-(benzenesulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
1-(1-benzoxepine-4-carbonyl)-3-(1H-imidazol-2-yl)piperidine
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
2-(3,4-dimethoxyphenyl)-1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
5-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
5-(3-fluoropropyl)-3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3R,9aR)-3-(2-methylpropyl)-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(1H-imidazol-1-ylmethyl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidine
3-fluoro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(pyridin-4-yl)quinoline
{1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
1-[4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
9-methoxy-7-oxo-3-[5-oxo-1-(propan-2-yl)pyrrolidine-3-carbonyl]-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-methyl-5-{[({[1-(4-methylphenyl)ethyl]carbamoyl}methyl)amino]methyl}furan-2-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-acetyl-8-[3-(1H-pyrazol-4-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-(6-chloroquinolin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
3-{[1-phenyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
3-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 4-{[(1-cycloheptyl-6-oxopiperidin-3-yl)formamido]methyl}benzoate
3-fluoro-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]acetamide
7-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
2-ethyl-4-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide
1-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]-3-methylbut-2-en-1-one
N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(4-fluorophenyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,4-diazepane
(3R,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-cyclopropyl-3-methylpiperidin-4-ol
(2S)-N-(3-chloro-4-propoxyphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
8-[(2-butyl-1H-imidazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylpyridine-3-carboxamide
1-[(4-methanesulfonylphenyl)methyl]-3-propoxypiperidine
4-[4-(3,5-dimethylphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
2,3-dimethyl-6-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-N-phenylpiperidine-1-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
N-{1-[2-(pyridin-2-yl)ethyl]-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1H-1,3-benzodiazol-7-yl}acetamide
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3-(2-methylpropyl)-1,2-oxazole
2-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-5,8-dimethylquinolin-4-ol
N-(4-ethylpyridin-2-yl)-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-hydroxypyridine-3-carboxamide
1-methyl-4-({4-[3-methyl-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)piperazine
3-(5-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-methylthiophene-2-carboxamide