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1,3-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-hexyl-8-(2-hydroxypyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(cyclopropylmethyl)-4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-6-methoxy-1,2-dihydroquinolin-2-one
3-ethyl-8-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-[2-(1H-imidazol-2-yl)benzoyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
2-(cyclohex-1-en-1-yl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}ethan-1-one
ethyl 5-(2,6-dimethylquinoline-4-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2R)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-2-phenylacetamide
(2S,4R)-4-amino-1-(isoquinoline-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
5-(4-fluorophenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-ol
2-chloro-N-(2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}ethyl)benzamide
7-(3,3,3-trifluoro-2-hydroxypropanoyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-(4-cyclohexylpiperazine-1-carbonyl)-1-[2-(3-fluorophenyl)ethyl]piperidin-2-one
(1S,5R)-N-(2-chloro-6-methylphenyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(piperazin-1-yl)ethan-1-one
{3-[(3-chlorophenyl)methyl]-1-(2,5-dimethylbenzenesulfonyl)piperidin-3-yl}methanol
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-(3-methoxyphenyl)piperidine
2-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-6-methylphenol
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-(but-2-yn-1-yl)-5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
2-methoxy-5-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]pyridine
N-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(2-fluorophenyl)methyl]piperidin-3-amine
5-[1-(4-fluorobenzoyl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-(3-chlorophenyl)-4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-[2-(4-phenylpiperidin-1-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(2-chloro-4-fluorobenzoyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-(4-hydroxyphenyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
(3S,4S)-1-(3,6-dimethylpyrazin-2-yl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-(1-methyl-1H-pyrrol-2-yl)-2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethane-1,2-dione
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
N4-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-6-methylpyrimidine-2,4-diamine
1-[4-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-[(2,6-difluorophenyl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[6-(trifluoromethyl)pyridin-2-yl]-decahydro-1,6-naphthyridin-2-one
3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
3-methanesulfonamido-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-methoxybenzamide
N-cyclopropyl-N-(3-phenylprop-2-yn-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-(2-fluorophenyl)-N-{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzamide
4-methyl-2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
6-(morpholin-4-yl)-N4-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrimidine-2,4-diamine
8-[3-(2,4-difluorophenyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-tert-butyl-4-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-(6-methoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide