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3-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazol-2-yl)pyridine
1-{3-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-[2-(cyclohex-1-en-1-yl)pyridine-4-carbonyl]morpholine
N-methyl-4-(piperidin-1-ylmethyl)-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
1-[2-hydroxy-5-(1H-pyrazol-3-yl)phenyl]ethan-1-one
1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-3-carboxamide
1-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-3-(1-methylpiperidin-4-yl)propan-1-one
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](quinolin-2-ylmethyl)amine
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
1-phenyl-4-(piperidin-3-yl)piperazine
N-({7-[(2-hydroxyphenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
[(2S,6S)-4-(1,3-benzothiazole-6-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
methyl 8-[(3,4-dimethoxyphenyl)methyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2-benzyl-1,3-thiazole-4-carbonyl)azepan-3-amine
2-(5-amino-4H-1,2,4-triazol-3-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-[1-(2-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
4-(morpholine-4-carbonyl)-1,2-dihydroisoquinolin-1-one
2-[(4-benzylpiperidin-1-yl)methyl]-3,5-difluoropyridine
N-(1-ethyl-5-oxopyrrolidin-3-yl)-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylpentanamide
5-ethyl-N-{2-[ethyl(methyl)amino]butyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-ethyl-4-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-[2-({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
2-amino-4-(2,2-dimethylpropyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
(1S,5R)-3-benzyl-6-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-1-cyclopentyl-4-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetamido]-N-ethylpyrrolidine-2-carboxamide
N-[4-(1-ethenyl-1H-pyrazol-4-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]-2,2-dimethylpropanamide
(4aR,7aS)-1-[2-(pyrrolidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-3-methyl-2-{[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}butanamide
{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methanamine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-amine
N-(2,3-dimethylphenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(2R,6R)-4-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-butyl-11-{[(2-chlorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
1-benzyl-4-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}pyrrolidin-2-one
2-(3-methoxyphenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
{[5-(3-fluoropyridin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-N-{1-oxaspiro[4.4]nonan-3-yl}piperidin-4-amine
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
5-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-benzyl-2-(4-{4-[(1,1-dioxo-1λ6-thiolan-3-yl)amino]piperidin-1-yl}phenyl)acetamide
ethyl 1-{2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetyl}piperidine-3-carboxylate
N'-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)ethanediamide
6-[4-(4-methylphenyl)benzoyl]-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
8-[(2-hydroxy-4-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione