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4-(4-fluoro-3-methylbenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-({[(2-benzyl-1,3-thiazol-4-yl)methyl]amino}methyl)pyrrolidin-3-ol
1-[4-({3-[2-hydroxy-3-(4-methyl-1,4-diazepan-1-yl)propoxy]-4-methoxyphenyl}methyl)piperazin-1-yl]ethan-1-one
N-(3-acetylphenyl)-3-{[methyl(oxan-4-yl)amino]methyl}benzamide
2-(5-chloro-2-ethoxyphenyl)-4-(pyrrolidine-1-carbonyl)pyridine
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
2-butyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
1-(1H-imidazol-2-ylmethyl)-5-[4-methoxy-3-(methoxymethyl)phenyl]-4-phenyl-1H-imidazole
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-[2-(pyrrolidin-1-yl)ethyl]piperidine
3-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]urea
N-{2-[5-methyl-4-({[(1R,2S)-2-propylcyclopropyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-3-carboxamide
4-cyclopentyl-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-3-methyl-1H-pyrazole-5-carboxamide
1-(pyridin-3-ylmethyl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}pyrrolidin-2-one
3-cyclopentyl-3-[(2,4-dimethoxyphenyl)methyl]-1-(4-methoxyphenyl)urea
(1R,5R)-3-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-[(2R,3R)-2-methoxy-1'-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
3-benzyl-4-(8-fluoroquinoline-2-carbonyl)piperazin-2-one
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(pentan-3-yl)piperidin-4-yl]acetate
6-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)oxane-4-carboxamide
5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-1-methylpiperidin-2-one
{1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
4-(4-methoxy-3-methylphenyl)-6-(morpholin-4-yl)pyrimidin-2-amine
6-(oxolan-3-yl)-2-(4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
methyl[(2-methylpyridin-4-yl)methyl]{[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}amine
N-(2H-1,3-benzodioxol-5-yl)-2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]acetamide
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-N-methylpyrimidin-2-amine
2-(2-aminoethyl)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]quinazolin-4-amine
2-(dimethylamino)-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(3aS,6aS)-5-[(3-chloro-2,6-difluorophenyl)methyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-(2,2-dimethyloxan-4-yl)-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
(3S,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-3-ol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-({8-[(1-methyl-1H-indol-3-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(trifluoromethyl)benzamide
4-[(4-fluorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,5R)-6-benzyl-3-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-(4-hydroxy-3-methoxybenzoyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
3,3-dimethyl-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
1,7-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-imidazole-5-carboxamide
2-{4-[2-(2,6-dimethoxyphenoxy)ethyl]-2-oxopiperazin-1-yl}benzonitrile
1-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-(pyridin-3-yl)ethane-1,2-dione
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}propanamide
{6-[2-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}methanol
1-methanesulfonyl-N-methyl-N-[2-(4-methylphenoxy)ethyl]piperidin-4-amine
4-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-methyl-1-benzofuran-7-carbonyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine