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6-chloro-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
(3S,4R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-N3-methyl-N5-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,3-dimethylphenoxy)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]acetamide
8-[(3,4-difluorophenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepan-5-one
2-amino-N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-4-methylpyrimidine-5-carboxamide
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
5-[4-(2-fluorophenyl)piperazin-1-yl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-(3-methoxypropyl)-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-[4-(dimethylamino)benzoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(8-methoxyquinolin-2-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-amino-6-(2,5-dimethylphenyl)-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-1-(propan-2-yl)piperidin-4-amine
2-ethyl-9-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(2,6-dimethoxyphenyl)-9-methoxy-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-4-(2-phenylethyl)piperazin-2-one
1-(2H-1,3-benzodioxole-5-carbonyl)-N-(3,4-difluorophenyl)piperidin-3-amine
3-(4-hydroxyphenyl)-2-phenyl-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
2-[2-(2-phenylphenyl)-1H-imidazol-1-yl]acetamide
5-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-2-(pyridin-2-yl)pyrimidine
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(propan-2-yloxy)ethyl]piperidine-4-carboxamide
N-[3-(1H-indol-1-yl)propyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(morpholin-4-yl)propanamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1-benzofuran-2-carboxamide
1-[4-(1H-imidazol-1-yl)benzoyl]-2-methyl-4-(2-methylphenyl)piperazine
3-methyl-4-(1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
5-[4-(2-amino-6-fluoro-1,3-benzothiazol-4-yl)phenyl]imidazolidine-2,4-dione
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]propanamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-[3-(4-hydroxyphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-(oxan-4-ylmethyl)acetamide
6-(2-chlorophenyl)-N-(1,4-dioxan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S,4R)-1-{[cyclohexyl(methyl)carbamoyl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl})amine
2-methoxy-N-[(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]oxolane-2-carboxamide
N-(2-methanesulfonamidoethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
4-methoxy-2-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
1-(1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
(1S,5R)-6-[4-(1H-imidazol-1-yl)benzoyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]propanamide
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(2-methylpyrimidin-4-yl)piperidine-4-carboxylic acid
4-{5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]furan-2-carbonyl}morpholine
[(3-chloropyridin-4-yl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
methyl (2S,4R)-1-(1-ethylpiperidin-4-yl)-4-[3-(3-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
(3R,4R)-4-cyclopropyl-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-methylpiperidin-4-ol
N-(2-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide