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5-{1-[1-(thiophen-2-yl)butyl]-1H-1,2,3-triazol-4-yl}pyrimidine
3-{[(2-ethylpyrimidin-4-yl)methyl](methyl)amino}-1-phenylpropan-1-ol
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-[1,3-dioxo-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(2-phenylethyl)piperidine-3-carboxamide
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
5-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
N-[(2R,3R)-1'-[(3-acetylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
4-chloro-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
4-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]azetidin-3-yl}morpholine
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
N-(2-chloro-5-sulfamoylphenyl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
2-propyl-N-[2-(4-sulfamoylphenyl)ethyl]-1,3-thiazole-4-carboxamide
1-(3-cyano-4-methoxyphenyl)-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
3-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[3-(trifluoromethyl)phenyl]ethyl}propanamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-acetamidopropanamide
(2R)-2-methyl-3-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]propan-1-ol
[3-(furan-3-carbonyl)-9-(pyridin-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
methyl 2-chloro-5-({2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carbonyl}amino)benzoate
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(pyridin-2-yl)acetamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
N-(1-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(thiophene-2-carbonyl)piperidine
3-cyano-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]benzamide
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,3-benzodiazole
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-ethyl-3-methylpiperidine-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylfuran-3-carboxamide
7-{2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
2-cyclohexyl-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-methyl-2-({1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
N-benzyl-N-(cyclopropylmethyl)-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
3-hydroxy-N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)benzamide
6-[2-(hydroxymethyl)phenyl]-4-methyl-1,2-dihydroquinolin-2-one
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methyl-3-[2-(methylsulfanyl)phenyl]urea
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]benzamide
N-[3-({[3-(2-oxopyrrolidin-1-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-(3-fluoro-5-methylphenyl)-3-[(2S)-pyrrolidin-2-ylmethyl]urea
N-methyl-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)-N-(quinolin-6-ylmethyl)propanamide
1-(diethylamino)-3-[2-methoxy-4-({[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-{4-[2-(4-fluoropiperidin-1-yl)-2-oxoethyl]phenyl}butanamide
2-{[5-(diphenylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-{[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
N-ethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyridazine-4-carboxamide
2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide