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4-[2-({4-benzyl-5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)ethyl]morpholine
(2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
6-methyl-4-[4-(pyrimidin-4-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(1s,4s)-4-hydroxy-N-[3-(pyridin-3-yloxy)propyl]cyclohexane-1-carboxamide
N-({5-[(2-methyl-1,3-oxazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
8-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[3-(morpholine-4-carbonyl)piperidin-1-yl]ethan-1-one
4-[4-(3-methyl-1-benzofuran-2-yl)-1H-1,2,3-triazol-1-yl]-1-propylpiperidine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
N-(2,2-dimethyloxan-4-yl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]morpholin-3-yl}-N-(2-fluorophenyl)acetamide
3-methyl-1-{1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}butan-1-ol
3,5-dichloro-4-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}pyridine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,3-difluoro-4-methylbenzamide
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1-(3-hydroxypyridine-2-carbonyl)-2-methyl-1,4-diazepan-5-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
1-(3-cyano-4-methylphenyl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
N-[(2,6-dimethoxyphenyl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
methyl 3-butanamido-6-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-methyl-1-benzofuran-2-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(3-methylbutanoyl)piperidine-3-carboxylate
1-benzyl-5-methanesulfonamido-2-methyl-N-[(6-methylpyridin-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
9-[2-(5-fluoro-2-methylphenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-3-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(3-phenylpropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(4-chloro-1H-pyrazol-1-yl)methyl]-1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazole
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methyl-1H-pyrazole
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[1-(methylsulfanyl)propan-2-yl]piperidine
1-(furan-2-ylmethyl)-N-(thiolan-3-yl)piperidine-4-carboxamide
5-acetyl-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]thiophene-2-carboxamide
2-{4-[(2-methoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{[3-methyl-7-(4-oxo-4-phenylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
diethyl({3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
(2R)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-methoxy-2-phenylacetamide
5-butyl-1'-(5-propyl-1,3,4-thiadiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-(2,3-dihydro-1-benzofuran-2-carbonyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[2-(furan-2-yl)azepane-1-carbonyl]-5-methoxy-1-methyl-1H-indole
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
N-[2-(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
(furan-3-ylmethyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-[(3-chlorophenyl)methyl]-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[3-(4-fluorophenoxy)propyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
ethyl 4-{methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}piperidine-1-carboxylate
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethan-1-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)acetamide
9-(2,4-difluorophenyl)-N,15-dimethyl-N-(1,2-oxazol-3-ylmethyl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-4-phenylbutanamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(pyrrolidine-1-carbonyl)pyridine