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4-[(3,4-dimethoxypyridin-2-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(cyclohexylmethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-(cyclopropylmethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
3-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(dimethylamino)-N-(1-{7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
5-methoxy-N-(2-methoxyethyl)-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
3-(4-chlorobenzoyl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
4-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,2-dihydroquinolin-2-one
4-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2-(methylsulfanyl)pyrimidine
4-[3-(2-methoxyphenyl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzene-1-sulfonamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]propanamide
2-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-ylmethyl)phenoxy]acetamide
methyl 8-[(4-fluorophenyl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
2-amino-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-ethyl-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-fluoro-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[2-(ethylsulfanyl)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
methyl 3-[(2-chloro-6-fluorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-[(diethylamino)methyl]-N-(pyrrolidin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[1-(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
3-chloro-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-({8-[(2-ethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
2,3-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-[4-(pyridin-3-yloxy)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-ethyl-5-methyl-4-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-oxazole
[(5-methoxy-1H-indol-2-yl)methyl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
3-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,6S)-4-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)-2,6-dimethylmorpholine
1-[(3,5-dimethylphenyl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
1-(2-chloro-5-methylphenyl)-3-[2-hydroxy-3-(pyrrolidin-1-yl)propyl]urea
(3S)-3-{[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]amino}azepan-2-one
4-(cyclopropylmethyl)-1-(5-fluoro-1H-indole-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
ethyl 4-[(4-chlorophenyl)methyl]-1-(furan-3-carbonyl)piperidine-4-carboxylate
N-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
N-(1-methanesulfonylpiperidin-4-yl)-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
2-(3,5-dimethoxybenzoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-methyl-2-oxo-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-{4-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
methyl N-[4-(2-amino-6-methylpyridin-3-yl)phenyl]carbamate
5-chloro-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
3-hexyl-8-(2-methoxypyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(azocan-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
1-[(4-methoxyphenyl)methyl]-4-(oxolane-3-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-cyclohexyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(5-{[6-(dimethylamino)pyrimidin-4-yl]amino}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
1-{2-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
2,5-dimethoxy-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide