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6-(benzyloxy)-4-[3-(2-chlorophenyl)propanoyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
N-[(1-ethylpiperidin-3-yl)methyl]-5-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
N-methyl-N-({1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)furan-2-carboxamide
3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
1-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1H-1,2,4-triazole
2-{4-cyclohexyl-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-butyl-5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-benzoxazole
3-(1H-imidazol-2-ylmethyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
1-methyl-3-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}-1,2-dihydroquinolin-2-one
2-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-1,2-dihydroisoquinolin-1-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[4-(1H-pyrazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl 8-[(3,4-difluorophenyl)methyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(2-fluorophenyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-5-carboxamide
4-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}phenol
6-methyl-2-[(2R)-oxolane-2-carbonyl]-5-[5-(pyridin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2-(2-phenylethyl)piperidine
methyl (2S,4S)-1-(2,2-diphenylethyl)-4-(3-hydroxynaphthalene-2-amido)pyrrolidine-2-carboxylate
4-[(3-hydroxyphenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(2H-1,3-benzodioxol-5-yl)-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(dimethyl-1,2-oxazol-4-yl)-N-(pyridin-3-ylmethyl)propanamide
2-cyclopropyl-3-oxo-N-[(1R)-1-phenylpropyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[3-(2,2-dimethylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
2-{4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperazin-1-yl}benzonitrile
N-[1-(1-benzothiophene-5-carbonyl)piperidin-4-yl]pyrimidin-2-amine
N-(azepan-2-ylmethyl)-5-ethyl-1,3,4-oxadiazol-2-amine
9-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
4-chloro-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-pyrazol-5-amine
1-cyclopentyl-5-(4-cyclopentylpiperazine-1-carbonyl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
3-[(3-fluorophenyl)methyl]-N-(3-phenylpropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[2-(ethanesulfonyl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(2-methoxyphenyl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
8-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(1-propylpiperidin-4-yl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}ethan-1-one
2-chloro-4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-imidazol-2-yl}phenol
4-(1-methyl-1H-imidazol-2-yl)-1-(3-phenylpropyl)piperidine
methyl 3-({[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate
3-[2-(2,4-difluorophenyl)ethyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
N-methyl-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidine-2-carboxamide
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-[(3-fluorophenyl)methyl]-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-ethyl-3-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
1-[3-(dimethylamino)phenyl]-3-[3-(methylsulfanyl)propyl]urea
N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]cyclohex-1-ene-1-carboxamide
3-methyl-1-[(3E)-4-methylhex-3-en-1-yl]-1,2-dihydroquinoxalin-2-one
N-[2-(2,4-difluorophenyl)-1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-methylpyridin-2-amine
4-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-ethylpiperazin-2-one