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5-[1-(cyclopropylmethyl)pyrrolidin-2-yl]-N-{2-[(pyridin-3-yl)amino]ethyl}thiophene-2-carboxamide
N-[3-(4-{[2-(2-fluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methoxyacetamide
5-(dimethylamino)-2-[2-(1-methylpiperidin-2-yl)ethyl]-2,3-dihydropyridazin-3-one
ethyl 4-[4-(4-{[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
3-cyclopropyl-N-[2-(5-methylthiophen-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-phenyl-4-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperazin-2-one
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
{4-methyl-5-[(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methyl]-4H-1,2,4-triazol-3-yl}methanol
3-(2-amino-1,3-thiazol-4-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(4-methoxyphenyl)prop-2-yn-1-one
3-(4-methylpiperazin-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]propanamide
5-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-N-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(2E)-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(thiophen-2-yl)prop-2-enamide
3-amino-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]acetamide
4-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1λ6-thiane-1,1-dione
(1-{1-[6-(2-methoxyphenyl)-3-(thiomorpholine-4-carbonyl)pyridin-2-yl]piperidin-4-yl}piperidin-3-yl)methanol
1-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-hexyl-8-(oxane-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)morpholine
3-(aminomethyl)-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
2-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
N-(2-methoxyethyl)-3-oxo-N-(thiophen-2-ylmethyl)-2,3-dihydro-1H-indene-1-carboxamide
3-methyl-8-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-phenyl-1-{4-[(2,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-4-{2-[2-(dimethylamino)ethoxy]phenyl}-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
(2R,3S,6R)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-(2-fluoro-5-methylphenoxy)-1-[(propan-2-yl)carbamoyl]piperidine-4-carboxylic acid
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(diphenylmethyl)propanamide
2-{[(1-benzylpyrrolidin-3-yl)(methyl)amino]methyl}pyridine-3-carboxylic acid
2-[3,5-dimethyl-4-(quinolin-6-yl)-1H-pyrazol-1-yl]acetic acid
2-(dimethylamino)-4-methyl-N-[2-(methylamino)ethyl]pyrimidine-5-carboxamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
3-(furan-2-ylmethyl)-1-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}urea
N-benzyl-3-(pyridin-3-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
6-({[2-(4-phenylpyrimidin-2-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
N-[(3S,4R)-1-(4-methyl-1H-imidazole-2-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-{[1-(4-fluorophenyl)cyclopropyl]methyl}piperidin-4-ol
3-(1-ethyl-1H-pyrazol-4-yl)-4-(2-ethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2,4-difluorophenoxymethyl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1,2-oxazole-3-carboxamide
3-(4-methoxyphenyl)-3-phenyl-1-(pyrrolidin-1-yl)propan-1-one
methyl 5-{[5-(oxan-2-yl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(3-methoxyphenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-one
5-(1-cyclohexanecarbonylpiperidin-4-yl)-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
7-(1,3-benzothiazol-2-yl)-4-(2,6-dimethoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-cyclohexyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}butanamide