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8-(2-amino-2-methylpropyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(cyclopropylmethyl)-2-[2-(2-methylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(2,5-dimethoxyphenyl)methyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-methylphenol
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-4-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butan-1-one
8-(2-hydroxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-amino-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
4-(2-chloro-4-fluorophenyl)-N-methylbenzamide
8-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[methyl({1H-pyrrolo[2,3-b]pyridin-6-yl})amino]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-(thiolan-3-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-(1,3-benzoxazol-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-{2-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
6-fluoro-2-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-fluorophenoxy)piperidine
methyl 1-[(4-{spiro[2.5]octane-1-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidine-4-carboxylate
ethyl 1-ethyl-5-[(4-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
(5S,9aS,9bS)-2-cyclopentyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1-benzothiophen-2-ylmethyl)-1-[2-(dimethylamino)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
N-({8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
2-(4-{[4-(furan-2-yl)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methoxy-4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
3-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
N-(cyclobutylmethyl)-2-methoxy-N-(oxolan-2-ylmethyl)quinoline-4-carboxamide
2-(4-methoxy-2-methylphenyl)-2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
5-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-[4-(azepan-1-yl)-3-chlorophenyl]-2-(morpholin-3-yl)acetamide
2-[(4aR,7aS)-4-(2-butoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[(3R,4S)-1-[(3-cyanophenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]cyclobutanecarboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
2-(1H-1,2,3,4-tetrazol-1-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-phenyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,2-diphenylacetamide
2-methyl-2-[(4-methylphenyl)amino]-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]propanamide
(3aR,6aR)-2-[2-(3-fluoro-4-methylphenyl)acetyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]urea
4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
4-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-phenylpropyl)morpholine
1-(azepane-1-sulfonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(2S)-2-hydroxy-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-phenylpropan-1-one
N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
2-methoxy-4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]quinoline
(2R)-2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}propanamide
N-[(2R,3R)-1'-(dimethyl-1,2-oxazole-4-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-{4-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-phenyl-1H-pyrazol-3-yl}pyridine