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1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-(4-methoxybenzoyl)piperazine
3-(1,3-benzothiazol-2-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(2-methoxyethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(3-hydroxypropyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
2-methyl-N-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}propanamide
2-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(piperidin-3-yl)benzamide
[(5-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
8-(5-methyl-1,3-oxazole-4-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(pyrimidin-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(cyclopropylmethyl)-5-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-cyclohexyl-4-(2-methylpyrrolidine-1-carbonyl)-1H-pyrazole
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-indol-1-yl)propan-2-yl]butanamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[3-(1H-imidazol-2-yl)benzoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N,N-bis(prop-2-en-1-yl)benzamide
5-chloro-4-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
N-(2,3-dihydro-1H-inden-1-yl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
5-(3,4-difluorophenoxymethyl)-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1R,2R,6S,7S)-N-[4-chloro-3-(ethylcarbamoyl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
2-[2-(5-cyclopropyl-1H-pyrazol-1-yl)ethyl]-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 4-[3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamido]piperidine-1-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}piperidin-2-one
methyl 3-{[(2-methyl-1,3-thiazol-4-yl)formamido]methyl}-5-(2-phenylacetamido)benzoate
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-methoxyphenyl)ethyl]propanamide
6-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-5-oxopentanamide
methyl 5-[(1-methoxypropan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}benzoic acid
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
(5S,9aS,9bS)-5-(3,4-difluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(3-{cyclopropyl[(2-methoxyphenyl)methyl]carbamoyl}phenyl)amino]acetic acid
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
2-{4-[(3-ethoxyphenyl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidin-2-yl)morpholine
3-methyl-3-[1-(1,2-oxazol-3-yl)ethyl]-1-[4-(propylsulfamoyl)phenyl]urea
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[3-(2-fluorophenoxy)azetidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
N-benzyl-1-cyclopentyl-N-ethyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-(methoxymethyl)-N-{[3-methyl-7-(2,4,5-trifluorobenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
1-tert-butyl-5-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
2-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-N-(3-methoxypropyl)-6-methylquinazolin-4-amine
4,6,7-trimethyl-2-{4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,4-diazepan-1-yl}quinazoline