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2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(pyrimidin-2-yl)phenol
3-methyl-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[1-(pyridin-2-yl)propan-2-yl]urea
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
(1S,5R)-6-{[4-(difluoromethoxy)phenyl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-1-benzyl-N-methyl-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
2-ethyl-8-(5-methyl-2-phenylfuran-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(1R,2S)-N-methyl-2-[4-(2-methylphenoxy)piperidine-1-carbonyl]cyclohexane-1-carboxamide
3-(azepane-1-carbonyl)-N-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,4S)-1,7,7-trimethyl-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-2-oxabicyclo[2.2.1]heptan-3-one
3-hydroxy-1-[(3-methylphenyl)methyl]-3-[(4-propylpiperazin-1-yl)methyl]piperidin-2-one
3-{2-oxo-2-[4-(quinazolin-4-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[(2-cyanophenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
4-butyl-11-(piperidin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}but-3-en-1-one
1'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-(3,5-dimethylfuran-2-carbonyl)-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(4-methyl-3-oxopiperazine-1-carbonyl)-3,4-dihydroquinazolin-4-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(5-methyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-ethyl-N-(2-methylprop-2-en-1-yl)propanamide
(1S,5R)-6-(cyclopropylmethyl)-3-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aS,7aR)-2-(2-cyclopentylacetyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-{[(diphenylmethyl)amino]methyl}-7-fluoro-1-(2-methylpropyl)-1,2-dihydroquinolin-2-one
{1-[7-chloro-2-(furan-2-yl)-8-methylquinoline-4-carbonyl]piperidin-4-yl}methanol
3-{4-[(2,3-difluoro-6-methoxyphenyl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
7-(5-chloropyridin-2-yl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-methoxypropyl)-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-4-phenyl-9-(1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1-benzofuran-5-carboxamide
4-(2-amino-6-methylpyrimidin-4-yl)-N-(1-cyclohexyl-1H-pyrazol-5-yl)piperazine-1-carboxamide
6-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
(2S)-3-(4-hydroxyphenyl)-2-{[4-methyl-2-(pyridin-3-yl)pyrimidin-5-yl]formamido}propanamide
N-[1-(1-cyclohexanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
N-[2-(dimethylsulfamoyl)ethyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
N4-methyl-N2-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-2,4-diamine
N-(4-fluorophenyl)piperidin-3-amine
2-{2-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-methyl-4-(4-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}phenyl)butan-2-ol
1-(3-phenylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]acetamide
2-methyl-4-{4-[3-(3-methylphenoxy)azetidine-1-carbonyl]phenyl}butan-2-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-hydroxybenzoyl)piperidin-3-ol
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-4-yl)acetamide
ethyl 3-({2-methyl-3-[(pyridin-3-ylmethyl)amino]phenyl}formamido)butanoate
(2S,4R)-4-{[(3,5-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-3-yl)pyridine