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3-(5-methylfuran-2-yl)-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[1-(1H-imidazol-1-yl)butan-2-yl]propanamide
2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)-4-{1-[1-(pyridin-3-yl)propan-2-yl]piperidin-3-yl}pyrimidine
(4aR,7aS)-1-cyclopropanecarbonyl-4-(thiophen-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}-N,N-dimethylpropanamide
N-cyclopentyl-4-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-4-oxobutanamide
ethyl 4-[4-(4-{[1-(thiophen-2-yl)propan-2-yl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
(2S,4S)-4-amino-N-ethyl-1-(2-methoxypyridine-4-carbonyl)pyrrolidine-2-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
(1R,2S)-2-[3-(carbamoylmethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-N-methylcyclohexane-1-carboxamide
methyl 2-{4-[(4-butyl-3-oxopiperazine-1-carbonyl)amino]phenoxy}acetate
N-[(3S,4R)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
5-acetyl-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-2-carboxamide
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
6-[(3-fluorophenyl)methoxy]-4-(furan-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-1H-indole
3-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
(3S,4S)-1-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-4-methylpiperidine-3,4-diol
2-({[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
2-(3-fluorophenyl)-N-(1-{4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
6-(2-ethoxyphenyl)-4-methyl-1,2-dihydroquinolin-2-one
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
6-[1-(7-chloroquinolin-4-yl)piperidin-3-yl]-2-methylpyrimidin-4-ol
(3S,5S)-1-butyl-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
N-[(1-methylpyrrolidin-3-yl)methyl]-7-(oxan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-({1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}methyl)propane-1-sulfonamide
7-[(2,5-dimethylphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-{4-[1-(2-ethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}propanamide
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-{[1-(cyclohexylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2-(5-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1-methyl-1H-imidazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-3-methyl-1H-pyrazole-4-sulfonamide
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(pyridin-3-yl)ethan-1-one
2-(5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}thiophen-2-yl)pyrrolidine
dimethyl(3-{2-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
3-benzyl-1-methyl-3-[2-oxo-2-(5-oxo-1,4-diazepan-1-yl)ethyl]-2,3-dihydro-1H-indol-2-one
1-(2,3-dichlorobenzoyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(2-phenylethyl)piperidin-4-yl)methanol
2-methoxy-N-[2-(quinolin-8-yl)phenyl]acetamide
3-[2-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
1-[(4-methoxyphenyl)methyl]-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazole
ethyl 3-(3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)propanoate
(3aR,7aS)-2-[2-(2-ethoxyethoxy)benzoyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
methyl 3-(furan-2-amido)-5-[(3-hydroxybutyl)amino]-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-methyl-4-[(6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]piperazine
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(pyrrolidin-3-yl)benzamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-2-carboxamide