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N,N-dimethyl-5-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)pyridin-2-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-4-(1H-pyrazol-4-yl)butan-1-one
1-cyclohexyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}piperidine-4-carboxamide
(3S,5R,9R)-11-[(3-fluoro-4-methylphenyl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-(oxolan-2-ylmethyl)-5-({3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyrimidin-2-amine
N-{[7-(3-chlorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-fluorobenzamide
5-(methoxymethyl)-N-[(1R,3S)-3-{[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}cyclopentyl]furan-2-carboxamide
2-[3-(dimethylamino)propyl]-9-(2-fluoro-2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-[2-(4-chlorophenyl)ethyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
N-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}methyl)pyridine-3-sulfonamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[2-(piperidin-1-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-methyl-6-{2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
2-{4-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]phenoxy}acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(1H-imidazol-1-ylmethyl)piperidine
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-fluorophenyl)ethan-1-one
3-[(oxan-2-ylmethyl)sulfamoyl]-N-(pyridin-3-yl)benzamide
1-[2-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)-N,N-bis(propan-2-yl)benzamide
2-(4-chloro-1H-pyrazol-1-yl)-N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]acetamide
N-(propan-2-yl)-4-({1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}amino)pyridine-2-carboxamide
3-[5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1,2,4-oxadiazol-3-yl]pyridazine
1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
(2E)-3-(3-fluorophenyl)-1-[7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]prop-2-en-1-one
N-(pyridin-2-ylmethyl)-2-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetamido]benzamide
1-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
2-[5-(6-methoxypyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-butyl-5-[(3-phenylpyrrolidin-1-yl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-3-(2-phenoxyacetyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-cyclopropanecarbonyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
1-(2-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(2-oxoazepan-1-yl)propanamide
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(piperidin-1-yl)propan-1-one
4,5-dimethyl 1-[(3S,5S)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5-[(quinolin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N-{[3-methyl-7-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
1-benzyl-3-(pyrrolidin-1-yl)piperidine
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
(2R,4S)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxypiperidine-2-carboxylic acid
1-(methoxymethyl)-N-[1-(4-methylbenzoyl)piperidin-4-yl]cyclobutane-1-carboxamide
2-(5-acetylthiophen-3-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]ethan-1-one
methyl 2-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}methyl)-1,3-oxazole-4-carboxylate
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]benzonitrile
5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-2,1,3-benzoxadiazole