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3-(3-chlorophenyl)-5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
(2R,4R)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxypyrrolidine-2-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
2-[({1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-3-yl}oxy)methyl]pyridine
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
methyl 2-[(2,3-dimethylphenyl)sulfamoyl]-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]-1-ethylpiperidine
4-(4-fluorophenyl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-oxobutanamide
6-methyl-5-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-(2H-1,2,3-benzotriazol-2-yl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
2-(azepan-1-yl)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}acetamide
1-[2-(1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
4-({4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
N-{4-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenyl}acetamide
(4aR,7aS)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(4-methoxyphenyl)-N-({1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}methyl)acetamide
3-methyl-1-{[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazol-5-amine
1-(2,3-dimethoxyphenyl)-2-(2-fluorobenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pentane-1,4-dione
2-({4-[(2-methoxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)benzonitrile
5-(furan-2-ylmethyl)-5-{3-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-N-(4-methoxyphenyl)piperidin-3-amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-4-yl)ethyl]acetamide
N-({7-cyclohexanecarbonyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
N-(6-cyanopyridin-3-yl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
ethyl 4-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperazine-1-carboxylate
2-ethyl-8-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aS)-1-oxo-5-(3-phenylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[2-oxo-2-(pyrrolidin-1-yl)ethyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
1-(4-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}phenyl)pyrrolidin-2-one
(1-methyl-1H-imidazol-2-yl)(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)methanol
1-cyclopentyl-3-(3-fluorophenyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amine
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenyl)piperidine
3-[(1-acetylpiperidin-4-yl)oxy]-N-[(3-fluorophenyl)methyl]-4-methoxybenzamide
{2-[2-(8-methoxyquinolin-2-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
(3S)-1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-ol
N-[(3R,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxyacetamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
3-(2H-1,3-benzodioxol-5-yl)pyridin-2-ol
6-{3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-N-{[4-(methylsulfanyl)phenyl]methyl}cyclopropanamine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
(3S,9aR)-3-(hydroxymethyl)-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
7-methyl-2-[2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione