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2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[1-(2-methylpropyl)cyclopropyl]acetamide
1-(2,3-dihydro-1-benzofuran-2-ylmethyl)-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methylurea
3-(2-cyclohexylacetyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
5-(2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
methyl (2S)-1-{6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carbonyl}pyrrolidine-2-carboxylate
2-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
3-(2-methoxyethyl)-1-[2-(3-methoxyphenoxy)ethyl]piperidine-3-carboxylic acid
{1-ethyl-5-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
5-{[2-(2-fluorophenyl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
N,N-dimethyl-2-{[2-(propylsulfanyl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-{[3-(furan-2-yl)phenyl]methyl}piperidine
N-{2-[4-(phenylcarbamoyl)-1H-1,2,3-triazol-1-yl]ethyl}pyridine-2-carboxamide
N-cyclohexyl-3-{4-[(phenylcarbamoyl)methyl]piperazin-1-yl}propanamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidine
3-[(dimethylamino)methyl]-1-(9H-purin-2-yl)piperidin-3-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2-(pyrrolidin-1-yl)propanamide
2-[3-(2-phenylethyl)-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl]pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}thiophene-2-carboxamide
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-{4-[2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamido]phenyl}pentanamide
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2-methoxy-6-methylphenyl)formamido]acetic acid
1-[1-(3-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-{1,3-dioxo-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
N-cyclopropyl-1-ethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
(3S,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3R,4R)-4-(morpholin-4-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
2-[5-(methoxymethyl)-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(piperidin-3-yl)benzamide
1-(2-chloroprop-2-en-1-yl)-7-fluoro-3-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-cyclobutanecarbonyl-3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidine
3-[1-(methoxymethyl)cyclopropyl]-1-[4-(2-methoxyphenyl)phenyl]-3-methylurea
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-2-ylsulfanyl)acetamide
[(2-fluoro-4-methoxyphenyl)methyl]({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
2-methyl-4-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}quinoline
1-ethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-cyclobutyl-3-{[1-(1H-imidazol-1-yl)butan-2-yl]sulfamoyl}benzamide
6-(4-ethylphenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-fluorophenyl)-N-[3-(3-hydroxypiperidin-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
4-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-2-methylphenol
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}acetamide
5-ethyl-N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
N-[2-(1H-imidazol-1-yl)ethyl]-4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-methylpyrimidin-2-amine
8-(5-fluoropyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one